Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataKi:  9.40nM ΔG°:  -46.6kJ/molepH: 6.0 T: 2°CAssay Description:Measurement of EP2 receptor binding affinity was carried out according to the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285 (...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 6(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  0.700nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  35nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 3(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  46.1nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  49.9nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 9(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  59nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 5(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  60nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 11(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  72nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 8(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  74.8nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 2(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  144nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 7(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  178nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistone deacetylase 4(Homo sapiens (Human))
Universidad Del PaíS Vasco

US Patent
LigandPNGBDBM119440(BDBM119696 | US8685986, 15)
Affinity DataIC50:  338nMT: 2°CAssay Description:The reactions were carried out in a 96-well microplate for fluorometry in a 50 μl reaction volume. After the deacetylation reaction, Fluor-de-Ly...More data for this Ligand-Target Pair
In DepthDetails US Patent