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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 23 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  8nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of recombinant full-length human HDAC6 expressed in baculovirus infected sf9 insect cells using Fluor de Lys as substrate preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of human HDAC6 using fluorogenic HDAC substrate incubated for 30 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  100nMAssay Description:Inhibition of human HDAC9 using fluorogenic HDAC substrate incubated for 30 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  100nMAssay Description:Inhibition of HDAC7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  100nMAssay Description:Inhibition of human HDAC7 using fluorogenic HDAC substrate incubated for 45 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  200nMAssay Description:Inhibition of HDAC9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  400nMAssay Description:Inhibition of HDAC5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  600nMAssay Description:Inhibition of HDAC4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human HDAC5 using fluorogenic HDAC substrate incubated for 30 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human HDAC8 using fluorogenic HDAC substrate incubated for 60 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Ghent University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human HDAC4 using fluorogenic HDAC substrate incubated for 30 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human HDAC11 using fluorogenic HDAC substrate incubated for 30 mins by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human HDAC2 using fluorogenic HDAC substrate incubated for 15 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human HDAC3 using fluorogenic HDAC substrate incubated for 10 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human HDAC10 using fluorogenic HDAC substrate incubated for 45 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human HDAC1 using fluorogenic HDAC substrate incubated for 15 mins by fluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of recombinant full length human HDAC1 expressed in Escherichia coli cells using Fluor de Lys as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of HDAC10 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of HDAC11 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50252392(CHEMBL4069287)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed