Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 13 hits in this display
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: <500nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: 750nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: 750nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: 7.50E+3nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
BDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
IC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair