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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

TargetHistone deacetylase 11(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50:  3nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 11(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50: <500nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 11(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50: <500nMAssay Description:The probe binding HDAC11 assay was performed using a time resolved fluorescence (TRF) assay format. Recombinant N-terminal GST tag full-length human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 8(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50:  750nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 6(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50:  750nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 7(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50:  7.50E+3nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 4(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 3(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 9(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 2(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 5(Homo sapiens (Human))
Forma Therapeutics

US Patent
LigandPNGBDBM421500(US10508088, Example 1-1 | US10508088, ID HDTK010 |...)
Affinity DataIC50: >1.00E+4nMAssay Description:This example describes in vitro inhibition properties of exemplary HDAC11 inhibitors for various HDACs. HDAC inhibition assays were performed using a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent