Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50306393(5-(4-(4-fluorophenoxy)benzyl)thiazolidine-2,4-dion...)
Affinity DataEC50:  500nMAssay Description:Partial agonist activity at human GPR40 expressed in CHO cells assessed as fatty acid-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50306393(5-(4-(4-fluorophenoxy)benzyl)thiazolidine-2,4-dion...)
Affinity DataEC50:  474nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50306393(5-(4-(4-fluorophenoxy)benzyl)thiazolidine-2,4-dion...)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human GPR40 by FLIPR assay in presence of 1% BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed