Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPoly(ADP-ribose) glycohydrolase(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL

LigandBDBM50350093(CHEMBL1813879)Copy SMILESCopy InChI

Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of PARG using [alpha-32P]ADP-ribose polymers after 5 mins by TRAP assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL

LigandBDBM50350093(CHEMBL1813879)Copy SMILESCopy InChI

Affinity DataIC50:  1.23E+5nMAssay Description:Inhibition of PARP-1 using [32P]-NAD+ after 15 minsMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathway
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI