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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetCarbonic anhydrase 6(Homo sapiens (Human))
Artvin£Oruh University

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataKi:  1.78E+4nMAssay Description:Inhibition of human carbonic anhydrase 6 esterase activity using 4-nitrophenylacetate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Artvin£Oruh University

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataKi:  2.15E+4nMAssay Description:Inhibition of human carbonic anhydrase 2 esterase activity using 4-nitrophenylacetate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Artvin£Oruh University

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of human carbonic anhydrase 4 esterase activity using 4-nitrophenylacetate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Artvin£Oruh University

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataKi:  3.51E+4nMAssay Description:Inhibition of human carbonic anhydrase 1 esterase activity using 4-nitrophenylacetate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
Jilin Province Academy Of Traditional Chinese Medicine And Materia Medica

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataIC50:  566nMAssay Description:Inhibition of human muscle recombinant aldose reductase by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataIC50:  680nMAssay Description:Inhibition of GST-tagged human recombinant PTB1B using pNPP as substrate after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Artvin£Oruh University

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataIC50:  3.83E+4nMAssay Description:Carbonic anhydrase activity was assayed by following the hydration of CO2 according to our previous studies [Soyut et al., Protein Pept. Lett., 15:52...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TCPTP after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 11(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of SHP2 using OMFP as substrate after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 6(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of SHP1 using OMFP as substrate after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase F(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50363494(5,5'-methylenebis(3,4,6-tribromo-benzene-1,2-d...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of LAR using OMFP as substrate after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed