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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi:  1.23nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-HT1A receptor in Sprague-Dawley albinus rat cerebral cortex membranes after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi:  36.7nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-HT1A receptor in Sprague-Dawley albinus rat cerebral cortex membranes after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]-5-CT from 5HT7 receptor in Sprague-Dawley albinus rat hypothalamic membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi:  299nMAssay Description:Displacement of [3H]-5-CT from 5HT7 receptor in Sprague-Dawley albinus rat hypothalamic membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-LY278584 from 5HT3 receptor in Sprague-Dawley albinus rat cerebral cortex membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-LY278584 from 5HT3 receptor in Sprague-Dawley albinus rat cerebral cortex membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]GR113808 from 5HT4 receptor in Sprague-Dawley albinus rat striatal membranes after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in Sprague-Dawley albinus rat striatal membranes after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley albinus rat frontal cortex membranes after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley albinus rat frontal cortex membranes after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]GR113808 from 5HT4 receptor in Sprague-Dawley albinus rat striatal membranes after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in Sprague-Dawley albinus rat striatal membranes after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359421(CHEMBL1926735)
Affinity DataEC50:  16.3nMAssay Description:Agonist activity at human 5HT1A receptor expressed in human HeLa cells assessed as inhibition of forskolin-stimulated cAMP production pretreated 20 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed