Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359430(CHEMBL1926757)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in Sprague-Dawley albinus rat striatal membranes after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359430(CHEMBL1926757)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-HT1A receptor in Sprague-Dawley albinus rat cerebral cortex membranes after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359430(CHEMBL1926757)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Sprague-Dawley albinus rat frontal cortex membranes after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(RAT)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359430(CHEMBL1926757)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-LY278584 from 5HT3 receptor in Sprague-Dawley albinus rat cerebral cortex membranes after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359430(CHEMBL1926757)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-5-CT from 5HT7 receptor in Sprague-Dawley albinus rat hypothalamic membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Universidad Complutense De Madrid

Curated by ChEMBL
LigandPNGBDBM50359430(CHEMBL1926757)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]GR113808 from 5HT4 receptor in Sprague-Dawley albinus rat striatal membranes after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed