Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 20 hits in this display
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
Ki: 422nMAssay Description:Competitive inhibition of recombinant human MAO-A using 0.01 to 0.5 mM kynuramine substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
IC50: 2.50E+3nMAssay Description:Inhibition of human recombinant MAOA using kynuramine as substrate preincubated for 30 mins followed by substrate additionMore data for this Ligand-Target Pair
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)
BDBM67454(1,2,4-trihydroxy-9,10-anthraquinone | 1,2,4-trihyd...)