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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetProcathepsin L(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM48563(2-phenyl-1H-quinolin-4-one | 2-phenyl-4-quinolone ...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human recombinant cathepsin L expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM48563(2-phenyl-1H-quinolin-4-one | 2-phenyl-4-quinolone ...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of human recombinant cathepsin V expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM48563(2-phenyl-1H-quinolin-4-one | 2-phenyl-4-quinolone ...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of tubulin polymerization(ITP)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEukaryotic translation initiation factor 4 gamma 1(Homo sapiens (Human))
Emory University

Curated by PubChem BioAssay
LigandPNGBDBM48563(2-phenyl-1H-quinolin-4-one | 2-phenyl-4-quinolone ...)
Affinity DataIC50:  6.40E+4nMAssay Description:Dose Response Confirmation for Small Molecule Inhibitors of Eukaryotic Translation Initiation NIH Molecular Libraries Screening Centers Network [MLSC...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay