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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetCarbonic anhydrase 2(Homo sapiens (Human))
Artvin Coruh University

LigandPNGBDBM50386171(CHEMBL253691 | hCA inhibitor, 5)
Affinity DataKi:  5.64E+3nMpH: 7.4Assay Description:CA activity was assayed by following the change in absorbance at 348 nm of 4-NPA to 4-nitrophenylate ion over a period of 3 min at 25°C using a spect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Artvin Coruh University

LigandPNGBDBM50386171(CHEMBL253691 | hCA inhibitor, 5)
Affinity DataKi:  5.64E+3nMAssay Description:Inhibition of human CA2 using 4NPA as substrate for 3 mins by Lineweaver burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Atat£Rk University

Curated by ChEMBL
LigandPNGBDBM50386171(CHEMBL253691 | hCA inhibitor, 5)
Affinity DataKi:  7.64E+3nMAssay Description:Inhibition of human CA4 using 4NPA as substrate for 3 mins by Lineweaver burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 6(Homo sapiens (Human))
Artvin Coruh University

LigandPNGBDBM50386171(CHEMBL253691 | hCA inhibitor, 5)
Affinity DataKi:  1.37E+4nMpH: 7.4Assay Description:CA activity was assayed by following the change in absorbance at 348 nm of 4-NPA to 4-nitrophenylate ion over a period of 3 min at 25°C using a spect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 6(Homo sapiens (Human))
Artvin Coruh University

LigandPNGBDBM50386171(CHEMBL253691 | hCA inhibitor, 5)
Affinity DataKi:  1.37E+4nMAssay Description:Inhibition of human CA6 using 4NPA as substrate for 3 mins by Lineweaver burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Artvin Coruh University

LigandPNGBDBM50386171(CHEMBL253691 | hCA inhibitor, 5)
Affinity DataKi:  1.84E+4nMpH: 7.4Assay Description:CA activity was assayed by following the change in absorbance at 348 nm of 4-NPA to 4-nitrophenylate ion over a period of 3 min at 25°C using a spect...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Artvin Coruh University

LigandPNGBDBM50386171(CHEMBL253691 | hCA inhibitor, 5)
Affinity DataKi:  1.84E+4nMAssay Description:Noncompetitive inhibition of human CA1 using 4NPA as substrate for 3 mins by Lineweaver burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed