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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 16 hits in this display   

TargetD(1A) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]-SCH-23390 from human dopamine D1 receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]-N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]-N-methylspiperone from human dopamine D2long receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity to adrenergic Alpha-2C receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  2.80E+3nMAssay Description:Binding affinity to dopamine D5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  3.50E+3nMAssay Description:Binding affinity to adrenergic alpha2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  6.40E+3nMAssay Description:Binding affinity to adrenergic alpha2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  1.80E+4nMAssay Description:Binding affinity to dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  1.30E+5nMAssay Description:Binding affinity to dopamine D3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  2.20E+5nMAssay Description:Binding affinity to 5HT7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  3.40E+5nMAssay Description:Binding affinity to adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  7.50E+5nMAssay Description:Binding affinity to dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  8.20E+5nMAssay Description:Binding affinity to adrenergic kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  8.70E+5nMAssay Description:Binding affinity to 5HT3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataKi:  2.65E+6nMAssay Description:Binding affinity to dopamine D4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50325822(CHEMBL1224527 | trans-(5R)-5-phenyl-1,2,3,4,4a,5,6...)
Affinity DataEC50:  0.640nMAssay Description:Agonist activity at human D1 receptor assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed