Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kJ/mol)

Found 2 hits in this display   

TargetHistone acetyltransferase p300(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

LigandBDBM50580969(CHEMBL5073432)Copy SMILESCopy InChI

Affinity DataIC50:  12nMAssay Description:Inhibition of p300 (unknown origin) preincubated for 15 mins followed by addition of substrate [3H] Ac-CoA and measured after 60 mins by liquid scint...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathway
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetCREB-binding protein(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL

LigandBDBM50580969(CHEMBL5073432)Copy SMILESCopy InChI

Affinity DataIC50:  51nMAssay Description:Inhibition of CBP (unknown origin) preincubated for 15 mins followed by addition of substrate [3H] Ac-CoA and measured after 60 mins by liquid scinti...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI