EVODIAMINE BDBM50366821
CHEMBL2171768 BDBM50016248 5-(Methylene)Evodiamine
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- Huang, G; Kling, B; Darras, FH; Heilmann, J; Decker, M Identification of a neuroprotective and selective butyrylcholinesterase inhibitor derived from the natural alkaloid evodiamine. Eur J Med Chem 81: 15-21 (2014)
- Wang, Z; Xiong, Y; Peng, Y; Zhang, X; Li, S; Peng, Y; Peng, X; Zhuo, L; Jiang, W Natural product evodiamine-inspired medicinal chemistry: Anticancer activity, structural optimization and structure-activity relationship. Eur J Med Chem 247: (2023)
- Wu, S; Huang, Y; Wang, T; Li, K; Lu, J; Huang, M; Dong, G; Sheng, C Evodiamine-Inspired Topoisomerase-Histone Deacetylase Dual Inhibitors: Novel Orally Active Antitumor Agents for Leukemia Therapy. J Med Chem 65: 4818-4831 (2022)
- Evo312: An Evodiamine Analog and Novel PKCĪ²I Inhibitor with Potent Antitumor Activity in Gemcitabine-Resistant Pancreatic Cancer.
- Wang, L; Fang, K; Cheng, J; Li, Y; Huang, Y; Chen, S; Dong, G; Wu, S; Sheng, C Scaffold Hopping of Natural Product Evodiamine: Discovery of a Novel Antitumor Scaffold with Excellent Potency against Colon Cancer. J Med Chem 63: 696-713 (2020)
- Wang, S; Yamamoto, S; Kogure, Y; Zhang, W; Noguchi, K; Dai, Y Partial Activation and Inhibition of TRPV1 Channels by Evodiamine and Rutaecarpine, Two Major Components of the Fruits of Evodia rutaecarpa. J Nat Prod 79: 1225-30 (2016)