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- ChEBML_146441 Receptor binding affinity towards opioid receptor delta
- ChEBML_146436 Affinity for opioid receptor delta sites
- ChEBML_147334 Affinity towards opioid receptor delta 1
- ChEBML_147340 Binding affinity for delta opioid receptor
- ChEMBL_664311 (CHEMBL1259346) Inhibition of delta opioid receptor
- ChEBML_145469 Antagonistic activity against Opioid receptor delta 1
- ChEBML_146728 Binding affinity towards Opioid receptor delta 1
- ChEBML_146780 Affinity against the Opioid receptor delta 1
- ChEBML_147138 Binding affinity against Opioid receptor delta 1
- ChEMBL_145487 (CHEMBL752130) Binding affinity for delta opioid receptor
- ChEMBL_146580 (CHEMBL755069) Agonistic activity for opioid receptor delta
- ChEMBL_147340 (CHEMBL756185) Binding affinity for delta opioid receptor
- ChEMBL_2437093 Inhibition of delta opioid receptor (unknown origin)
- ChEMBL_325674 (CHEMBL863228) Agonistic activity at delta opioid receptor
- ChEMBL_325927 (CHEMBL869397) Inhibition of human delta opioid receptor
- ChEMBL_329931 (CHEMBL868792) Binding affinity to Delta opioid receptor
- ChEMBL_366644 (CHEMBL864704) Binding affinity to delta opioid receptor
- ChEMBL_437131 (CHEMBL906528) Binding affinity to delta opioid receptor
- ChEMBL_459305 (CHEMBL926464) Binding affinity to delta opioid receptor
- ChEMBL_497293 (CHEMBL995855) Binding affinity to delta opioid receptor
- ChEMBL_556745 (CHEMBL959808) Binding affinity to delta opioid receptor
- ChEMBL_556766 (CHEMBL961464) Binding affinity at delta opioid receptor
- ChEMBL_589795 (CHEMBL1051418) Binding affinity to delta opioid receptor
- ChEMBL_598546 (CHEMBL1043538) Inhibition of delta-type opioid receptor
- ChEMBL_629560 (CHEMBL1120978) Binding affinity to delta opioid receptor
- ChEMBL_799949 (CHEMBL1941655) Binding affinity to delta opioid receptor
- ChEMBL_884329 (CHEMBL2210362) Binding affinity to delta opioid receptor
- ChEMBL_2033541 (CHEMBL4687699) Inhibition of delta-type opioid receptor receptor (unknown origin)
- ChEBML_147338 Binding affinity to cloned Opioid receptor delta 1
- ChEBML_1552634 Binding affinity at delta opioid receptor (unknown origin)
- ChEBML_1651394 Binding affinity to delta opioid receptor (unknown origin)
- ChEMBL_145056 (CHEMBL753990) Agonist activity for Opioid receptor delta 1
- ChEMBL_1452453 (CHEMBL3362477) Binding affinity to human delta opioid receptor
- ChEMBL_145311 (CHEMBL751917) Agonistic activity towards Opioid receptor delta 1
- ChEMBL_1453328 (CHEMBL3366612) Binding affinity to human delta opioid receptor
- ChEMBL_145765 (CHEMBL752783) Binding affinity against Opioid receptor delta 1
- ChEMBL_146728 (CHEMBL753266) Binding affinity towards Opioid receptor delta 1
- ChEMBL_147335 (CHEMBL756180) Binding affinity against Opioid receptor delta 1
- ChEMBL_2494534 Binding affinity to delta-opioid receptor (unknown origin)
- ChEMBL_302679 (CHEMBL839442) Binding affinity for human Delta opioid receptor
- ChEMBL_320775 (CHEMBL884730) Affinity towards cloned Opioid receptor delta 1
- ChEMBL_512434 (CHEMBL980775) Displacement of radioligand from delta opioid receptor
- ChEMBL_664949 (CHEMBL1259781) Binding affinity to human delta opioid receptor
- ChEMBL_771176 (CHEMBL1837093) Agonist activity at delta-type opioid receptor
- ChEMBL_856830 (CHEMBL2163095) Binding affinity to rat delta opioid receptor
- ChEMBL_146347 (CHEMBL873930) The compound tested for agonistic activity against [3H]- NT1 (Opioid receptor delta 1) opioid receptor
- ChEBML_146444 Compound was evaluated for the opioid receptor delta affinity
- ChEBML_147336 Displacement of [3H]DADLE from Opioid receptor delta 1
- ChEBML_147337 Binding affinity for Opioid receptor delta 1 was determined
- ChEBML_147341 In vitro binding affinity towards opioid receptor delta 1
- ChEBML_53586 Ability to displace [3H]DADL from delta opioid receptor
- ChEMBL_1283875 (CHEMBL3106326) Binding affinity to delta opioid receptor (unknown origin)
- ChEMBL_1339709 (CHEMBL3243304) Binding affinity to delta opioid receptor (unknown origin)
- ChEMBL_145325 (CHEMBL750413) Binding affinity at cloned human delta-opioid receptor
- ChEMBL_146322 (CHEMBL757531) Displacement of [3H]DADLE at delta-opioid receptor
- ChEMBL_146328 (CHEMBL757536) Binding affinity was measured on delta opioid receptor
- ChEMBL_147343 (CHEMBL756188) Opioid receptor delta 1 agonist activity was determined
- ChEMBL_1504510 (CHEMBL3590952) Antagonist activity against delta opioid receptor (unknown origin)
- ChEMBL_1504517 (CHEMBL3590959) Binding affinity to delta opioid receptor (unknown origin)
- ChEMBL_1507469 (CHEMBL3599494) Binding affinity to delta opioid receptor (unknown origin)
- ChEMBL_1539083 (CHEMBL3738444) Binding affinity to delta opioid receptor (unknown origin)
- ChEMBL_1552634 (CHEMBL3762573) Binding affinity at delta opioid receptor (unknown origin)
- ChEMBL_1869949 (CHEMBL4371116) Binding affinity to delta opioid receptor (unknown origin)
- ChEMBL_2128136 (CHEMBL4837565) Binding affinity to delta-opioid receptor (unknown origin)
- ChEMBL_327761 (CHEMBL870569) Displacement of [3H]DPDPE from delta opioid receptor
- ChEMBL_379861 (CHEMBL864849) Displacement of [3H]DPDE from delta opioid receptor
- ChEMBL_401406 (CHEMBL870425) Activity at delta opioid receptor by MVD assay
- ChEMBL_439695 (CHEMBL888806) Displacement of [3H]DADLE from delta opioid receptor
- ChEMBL_466558 (CHEMBL935650) Displacement of [3H]DADLE from opioid delta receptor
- ChEMBL_486183 (CHEMBL1013977) Displacement of [3H]DPDPE from delta opioid receptor
- ChEMBL_525305 (CHEMBL968094) Displacement of [125]OXY from delta opioid receptor
- ChEMBL_745569 (CHEMBL1775886) Displacement of [3H]DADLE from delta opioid receptor
- ChEMBL_963011 (CHEMBL2390019) Binding affinity to delta opioid receptor (unknown origin)
- ChEMBL_968736 (CHEMBL2399172) Binding affinity to delta opioid receptor (unknown origin)
- ChEMBL_146781 (CHEMBL754443) Opioid receptor affinity against the Opioid receptor delta 1 by using the curve-fitting program LIGAND
- ChEBML_146726 Binding affinity against delta opioid receptor from calf frontal cortex.
- ChEBML_146889 Ability to displace [3H]-deltorphin II from delta opioid receptor
- ChEBML_1573819 Inhibition of delta opioid receptor (unknown origin) by PDSP assay
- ChEBML_305941 Inhibitory concentration against Delta opioid receptor of mouse vas deferens
- ChEMBL_145192 (CHEMBL754437) Binding affinity towards delta-opioid receptor from CHO cells
- ChEMBL_145323 (CHEMBL750411) Inhibition of ligand binding to human delta opioid receptor.
- ChEMBL_145340 (CHEMBL750575) Inverse agonist potency at cloned human delta-opioid receptor
- ChEMBL_145631 (CHEMBL753544) Displacement of [3H]-naloxone from Opioid receptor delta 1
- ChEMBL_145904 (CHEMBL750393) Opioid receptor delta 1 agonism in mouse vas deferens
- ChEMBL_146340 (CHEMBL753789) Inhibition against delta-opioid receptor using [3H]DPDPE radioligand.
- ChEMBL_146437 (CHEMBL757334) Binding affinity was measured on opioid receptor delta sites.
- ChEMBL_146762 (CHEMBL755206) Binding affinity for rat brain Opioid receptor delta 1
- ChEMBL_147329 (CHEMBL756174) Binding affinity towards Opioid receptor delta 1 was evaluated
- ChEMBL_147339 (CHEMBL756184) Binding affinity towards Opioid receptor delta 1 was determined
- ChEMBL_1517222 (CHEMBL3620206) Displacement of [3H] DAMGO from human delta opioid receptor
- ChEMBL_1549028 (CHEMBL3756647) Displacement of [3H]DPDPE from human delta opioid receptor
- ChEMBL_1721385 (CHEMBL4136385) Binding affinity to delta-type opioid receptor (unknown origin)
- ChEMBL_302811 (CHEMBL839501) Binding affinity for delta opioid receptor of rat brain
- ChEMBL_302899 (CHEMBL830360) Inhibition of [3H]DPDPE binding to delta-Opioid receptor
- ChEMBL_327765 (CHEMBL871139) Activity at delta opioid receptor in mouse vas deferens
- ChEMBL_361576 (CHEMBL870153) Displacement of [125I]IOXY from human delta opioid receptor
- ChEMBL_401403 (CHEMBL855304) Displacement of [3H]DPDPE from human delta opioid receptor
- ChEMBL_449625 (CHEMBL898720) Displacement of [3H]deltorphin 2 from delta opioid receptor
- ChEMBL_53586 (CHEMBL665474) Ability to displace [3H]DADL from delta opioid receptor
- ChEMBL_647571 (CHEMBL1217618) Displacement of [3H]DPDPE from human delta opioid receptor
- ChEMBL_145474 (CHEMBL751261) Binding affinity determined against Opioid receptor delta 1 from human cloned receptor
- ChEBML_145899 Inhibitory potency against delta Opioid receptor delta 1 in longitudinal muscle preparation of mouse vas deferens
- ChEBML_146442 Compound was evaluated for the binding affinity to opioid receptor delta
- ChEBML_146451 In vitro opioid receptor delta mediated mouse vas deferens (MVD) assay
- ChEBML_146592 Displacement of [3H]DSLET from rat brain membrane opioid receptor delta
- ChEBML_146923 Binding affinity to delta opioid receptor was measured using [3H]DADLE
- ChEBML_217856 Compound was evaluated for the binding affinity to delta opioid receptor
- ChEBML_53430 Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligand
- ChEBML_53571 Binding affinity towards opioid Delta receptor using [3H]DADLE as radioligand
- ChEMBL_1335004 (CHEMBL3239391) Displacement of [3H]DPDPE from delta opioid receptor (unknown origin)
- ChEMBL_1353488 (CHEMBL3269824) Agonist activity at delta opioid receptor in mouse vas deferens
- ChEMBL_1365290 (CHEMBL3292384) Displacement of [3H]DPDPE from delta-opioid receptor (unknown origin)
- ChEMBL_145341 (CHEMBL750576) Inverse agonist potency at cloned human opioid receptor delta 1
- ChEMBL_145889 (CHEMBL754255) Inhibitory activity against Opioid receptor delta 1 using [3H]DPDPE
- ChEMBL_146339 (CHEMBL753788) Inhibition against Opioid receptor delta 1 using [3H]DPDPE radioligand.
- ChEMBL_147342 (CHEMBL756187) Inhibition of [3H]- diprenorphine binding to Opioid receptor delta 1
- ChEMBL_1552794 (CHEMBL3760687) Agonist activity at delta-opioid receptor in mouse vas deferens
- ChEMBL_1823727 (CHEMBL4323491) Displacement of [3H] diprenorphine from delta opioid receptor (unknown origin)
- ChEMBL_1906936 (CHEMBL4409294) Inhibition of delta opioid receptor (unknown origin) by MVD assay
- ChEMBL_325357 (CHEMBL861057) Functional bioactivity against delta opioid receptor in mouse vas deferens
- ChEMBL_326438 (CHEMBL867596) Agonistic activity at delta opioid receptor in mouse vas deferens
- ChEMBL_326603 (CHEMBL863384) Agonistic activity at delta opioid receptor in mouse vas deferens
- ChEMBL_328876 (CHEMBL859855) Displacement of [3H]DPDPE from cloned human delta opioid receptor
- ChEMBL_333515 (CHEMBL866454) Displacement of [3H]diprenorphine from human cloned delta opioid receptor
- ChEMBL_334062 (CHEMBL861271) Agonist activity at delta opioid receptor in mouse vas deferens
- ChEMBL_364004 (CHEMBL860182) Functional bioactivity against delta opioid receptor in mouse vas deferens
- ChEMBL_428453 (CHEMBL918954) Displacement of [3H]DSLET from rat brain delta opioid receptor
- ChEMBL_428456 (CHEMBL918957) Agonist activity at delta opioid receptor in mouse vas deferens
- ChEMBL_439348 (CHEMBL887341) Agonist activity at delta opioid receptor in mouse vas deferens
- ChEMBL_446659 (CHEMBL896954) Displacement of [3H]DPDPE from human cloned delta opioid receptor
- ChEMBL_447456 (CHEMBL896479) Displacement of [3H]DPDPE from cloned human delta opioid receptor
- ChEMBL_455040 (CHEMBL887069) Displacement of [3H]diprenorphine from human cloned delta opioid receptor
- ChEMBL_455045 (CHEMBL887074) Agonist activity at delta opioid receptor in mouse vas deferens
- ChEMBL_457568 (CHEMBL922768) Displacement of [3H]p-Cl-DPDPE from delta opioid receptor
- ChEMBL_477640 (CHEMBL928102) Agonist activity at delta opioid receptor in mouse vas deferens
- ChEMBL_543174 (CHEMBL1015122) Binding affinity to delta opioid receptor in rat brain membrane
- ChEMBL_607041 (CHEMBL1074669) Antagonist activity at delta opioid receptor by GTPgammaS bunding assay
- ChEMBL_615881 (CHEMBL1102715) Antagonist activity at delta opioid receptor in mouse vas deferens
- ChEMBL_647236 (CHEMBL1217377) Agonist activity at delta opioid receptor in mouse vas deference
- ChEMBL_749290 (CHEMBL1785225) Agonist activity at delta opioid receptor in mouse vas deference
- ChEMBL_876446 (CHEMBL2187198) Binding affinity to delta opioid receptor by radioligand binding assay
- ChEMBL_878565 (CHEMBL2188650) Agonist activity at delta opioid receptor in mouse vas deferens
- ChEMBL_882180 (CHEMBL2215453) Agonist activity at delta opioid receptor in mouse vas deferens
- ChEMBL_959948 (CHEMBL2383890) Displacement of [3H]DADLE from delta opioid receptor (unknown origin)
- ChEMBL_969758 (CHEMBL2404100) Agonist activity at delta opioid receptor in mouse vas deferens
- ChEBML_146581 Binding ability towards opioid receptor delta expressed in homogenates of rat brain.
- ChEBML_146597 Binding affinity against opioid receptor delta in rats by displacing [3H]DPDPE
- ChEBML_146725 Inhibitory activity against Opioid receptor delta 1 binding to bovine striatal membrane
- ChEBML_147018 Binding affinity against Opioid receptor delta 1 in guinea pig brain membranes
- ChEBML_147185 Inhibition of [3H]DTLET binding torat brain membrane Opioid receptor delta 1
- ChEBML_305139 In vitro agonist activity against Opioid receptor delta in mouse vas deferens
- ChEMBL_145072 (CHEMBL754003) Binding affinity towards delta-2 opioid receptor in guinea pig brain
- ChEMBL_145181 (CHEMBL754281) Binding affinity against delta-opioid receptor in guinea pig brain membranes
- ChEMBL_145189 (CHEMBL754289) Binding affinity against Opioid receptor delta 1 expressed on CHO cells
- ChEMBL_145314 (CHEMBL751920) Maximum percentage effect of standard Opioid receptor delta 1 (Cl-DPDPE)
- ChEMBL_145498 (CHEMBL752140) In vitro potency was measured against human Opioid receptor delta 1
- ChEMBL_145630 (CHEMBL857860) Inhibition of deltorphin II binding to human Opioid receptor delta 1
- ChEMBL_145894 (CHEMBL873615) Inhibitory concentration against delta opioid receptor in mouse vas deferens assay
- ChEMBL_145905 (CHEMBL750394) Tested for agonist activity against delta opioid receptor mouse vas deferens
- ChEMBL_1459558 (CHEMBL3369358) Binding affinity to human delta opioid receptor expressed in CHO cells
- ChEMBL_146647 (CHEMBL754931) Displacement of [3H]DSLET from rat brain membrane delta opioid receptor
- ChEMBL_147059 (CHEMBL754879) Displacement of [3H]DPDPE (0.63 nM) from Opioid receptor delta 1
- ChEMBL_147136 (CHEMBL754168) Binding affinity against Delta Opioid receptor in Guinea pig brain membranes
- ChEMBL_147146 (CHEMBL754178) Binding affinity towards delta-1 opioid receptor in guinea pig brain
- ChEMBL_1869951 (CHEMBL4371118) Activation of delta opioid receptor (unknown origin) expressed in CHO cells
- ChEMBL_1906935 (CHEMBL4409293) Inhibition of delta opioid receptor (unknown origin) by radioligand binding assay
- ChEMBL_2297275 Binding affinity to delta opioid receptor (unknown origin) assessed as inhibition constant
- ChEMBL_2331268 Binding affinity to delta opioid receptor (unknown origin) assessed as inhibition constant
- ChEMBL_303251 (CHEMBL826377) Inhibition of [3H]naltrindole binding to human Opioid receptor delta 1
- ChEMBL_305844 (CHEMBL829585) In vitro inhibition of opioid receptor delta using mouse vas deferens
- ChEMBL_312682 (CHEMBL833129) Agonistic activity against delta opioid receptor of mouse vas deferens assay
- ChEMBL_334075 (CHEMBL867136) Binding affinity at human delta opioid receptor expressed in CHO cells
- ChEMBL_349385 (CHEMBL863860) Displacement of [3H]DPDPE from delta opioid receptor in rat brain
- ChEMBL_366648 (CHEMBL865970) Agonist activity at delta opioid receptor by mouse vas deferens assay
- ChEMBL_423422 (CHEMBL911097) Activity at delta opioid receptor in ICR mouse by MVD assay
- ChEMBL_540961 (CHEMBL1030681) Displacement of [125I]deltorphin 2 from human cloned delta opioid receptor
- ChEMBL_594991 (CHEMBL1039849) Binding affinity to human delta opioid receptor expressed in CHO cells
- ChEMBL_813972 (CHEMBL2020484) Displacement of [3H]U-69,593 from mouse brain delta opioid receptor
- ChEMBL_830315 (CHEMBL2060904) Displacement of [3H]DPDPE from delta opioid receptor in mouse cerebellum
- ChEMBL_972358 (CHEMBL2412183) Antagonist activity at delta opioid receptor in ICR mouse vas deferens
- ChEMBL_146919 (CHEMBL757507) Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assay
- ChEMBL_145747 (CHEMBL752636) Effective concentration was measured towards delta opioid receptor using mouse vas deferens(MVD, delta) bioassay in vitro
- ChEMBL_147023 (CHEMBL753664) Binding affinity against delta Opioid receptor delta 1 using [3H]DADLE as radioligand in guinea pig brain
- ChEBML_146773 Opioid receptor binding affinity in rat brain membrane preparations by the displacement of [3H]- DPDPE (Opioid receptor delta 1-selective radioligand)
- ChEMBL_145480 (CHEMBL752896) Binding affinity for opioid receptor type, human Opioid receptor delta 1 expressed in membrane homogenates of COS-1 or CHO cells
- ChEMBL_146773 (CHEMBL755216) Opioid receptor binding affinity in rat brain membrane preparations by the displacement of [3H]- DPDPE (Opioid receptor delta 1-selective radioligand)
- ChEMBL_146774 (CHEMBL755217) Opioid receptor binding affinity in rat brain membrane preparations by the displacement of [3H]DSLET (Opioid receptor delta 1-selective radioligand)
- ChEBML_147028 Binding affinity of Opioid receptor delta 1 by the displacement of delta-selective [3H]DSLET from brain membrane preparations.
- ChEBML_145063 Compound was evaluated for its inhibitory activity against the Opioid receptor delta 1
- ChEBML_145327 Binding affinity towards Opioid receptor delta 1 by the displacement of [125I]-Deltorphin
- ChEBML_145891 Inhibitory activity against delta-opioid receptor in mouse vas deferens preparation using DADLE
- ChEBML_145901 Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assay
- ChEBML_146431 In vitro binding activity against opioid receptor delta using [3H]DPDPE) as radioligand
- ChEBML_146595 Inhibition of [3H]- ]DSLET binding to opioid receptor delta from rat brain membrane
- ChEBML_147037 Inhibition of [3H]DSLET binding to rat brain membrane Opioid receptor delta 1
- ChEBML_53570 inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenates
- ChEMBL_1337149 (CHEMBL3240180) Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes
- ChEMBL_1353485 (CHEMBL3269821) Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes
- ChEMBL_145065 (CHEMBL753996) Tested for binding activity against delta opioid receptor using [3H]naltridole ligand
- ChEMBL_145191 (CHEMBL754436) Binding affinity towards Opioid receptor delta 1 using [3H]DPDPE as radioligand
- ChEMBL_145196 (CHEMBL756059) Agonist potency using GTP-gamma [35S]- binding assay for delta-opioid receptor
- ChEMBL_145332 (CHEMBL750420) Binding affinity was measured against mutated human Opioid receptor delta 1 (W248L)
- ChEMBL_1456842 (CHEMBL3367575) Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes
- ChEMBL_145771 (CHEMBL752789) Inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD)
- ChEMBL_145902 (CHEMBL750391) Inhibitory potency against Opioid receptor delta 1 in mouse vas deferens assay
- ChEMBL_146432 (CHEMBL757183) In vitro binding activity against opioid receptor delta using [3DPDPE] as radioligand
- ChEMBL_146474 (CHEMBL882767) Antagonist activity against Opioid receptor delta 1 in mouse vas deferens assay
- ChEMBL_146586 (CHEMBL754820) Displacement of [3H]- DPDPE from delta opioid receptor in rat brain membrane
- ChEMBL_146587 (CHEMBL754821) Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane
- ChEMBL_146752 (CHEMBL753332) Inhibition of [3H]- DADLE binding to Rat brain Opioid receptor delta 1
- ChEMBL_146896 (CHEMBL751670) Affinity of [H]DADLE to the delta opioid receptor from rat brain
- ChEMBL_146908 (CHEMBL751121) Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPE
- ChEMBL_146921 (CHEMBL757313) Binding affinity for delta opioid receptor by displacing [3H]DADL was determined
- ChEMBL_146995 (CHEMBL753816) Inhibitory concentration was determined against delta-opioid receptor using [3H]- DPDPE radioligand
- ChEMBL_147018 (CHEMBL756220) Binding affinity against Opioid receptor delta 1 in guinea pig brain membranes
- ChEMBL_147031 (CHEMBL753672) Binding affinity towards Opioid receptor delta 1 using [3H]DADLE as radioligand.
- ChEMBL_147289 (CHEMBL755877) The binding affinity on delta-opioid receptor using [3H]- DPDPE as radioligand
- ChEMBL_1552640 (CHEMBL3762579) Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane
- ChEMBL_1897424 (CHEMBL4399459) Agonist activity at delta opioid receptor (unknown origin) expressed in CHO cells
- ChEMBL_303226 (CHEMBL827191) Inhibition of [3H][Ile5,6]-deltorphin I binding to rat Opioid receptor delta
- ChEMBL_303398 (CHEMBL840061) Inhibition of [3H]naloxone binding to rat brain homogenate Opioid receptor delta
- ChEMBL_305139 (CHEMBL832434) In vitro agonist activity against Opioid receptor delta in mouse vas deferens
- ChEMBL_305867 (CHEMBL831911) In vitro agonistic activity against opioid receptor delta of mouse vas deferens
- ChEMBL_310403 (CHEMBL833181) Inhibition of delta opioid receptor mediated GTPgammaS binding to CHO cell membranes
- ChEMBL_372755 (CHEMBL871099) Displacement of [3H]DDPDE from delta opioid receptor expressed in HEK293 cells
- ChEMBL_377408 (CHEMBL867956) Displacement of [3H]DPDPE from delta opioid receptor in Wistar rat brain
- ChEMBL_387796 (CHEMBL865494) Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane
- ChEMBL_425713 (CHEMBL913695) Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane
- ChEMBL_435626 (CHEMBL903983) Displacement of [3H]DPDPE from delta opioid receptor in rat brain membrane
- ChEMBL_443503 (CHEMBL892731) Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membrane
- ChEMBL_458379 (CHEMBL941713) Displacement of [3H]naltrindole from delta opioid receptor expressed in CHO cells
- ChEMBL_462212 (CHEMBL945981) Displacement of [3H]naltrindole from delta opioid receptor in rat brain membranes
- ChEMBL_462213 (CHEMBL945982) Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes
- ChEMBL_470713 (CHEMBL934554) Binding affinity to delta opioid receptor in Sprague-Dawley rat brain membrane
- ChEMBL_477636 (CHEMBL928098) Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membrane
- ChEMBL_534601 (CHEMBL989026) Displacement of [3H]diprenorphine from human delta opioid receptor in CHO cells
- ChEMBL_534710 (CHEMBL982799) Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane
- ChEMBL_556446 (CHEMBL955663) Displacement of [3H]DAMGO from delta opioid receptor in rat brain membrane
- ChEMBL_556843 (CHEMBL964703) Displacement of [3H]DPDPE from delta opioid receptor in rat brain membrane
- ChEMBL_563751 (CHEMBL993514) Displacement of [3H]NTI from delta opioid receptor expressed in CHO cells
- ChEMBL_575378 (CHEMBL1027052) Displacement of [3H]DADLE from delta opioid receptor in rat cerebellum membrane
- ChEMBL_591861 (CHEMBL1045065) Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane
- ChEMBL_592554 (CHEMBL1046761) Binding affinity to rat delta opioid receptor expressed in rat C6 cells
- ChEMBL_595271 (CHEMBL1043623) Agonist activity at human delta opioid receptor by [35S]GTPgammaS binding assay
- ChEMBL_611745 (CHEMBL1074339) Displacement of [3H]DADLE from delta opioid receptor expressed in CHO cells
- ChEMBL_612211 (CHEMBL1074149) Displacement of [3H]DPDPE from delta opioid receptor in rat brain homogenate
- ChEMBL_627498 (CHEMBL1111784) Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane
- ChEMBL_701347 (CHEMBL1648967) Displacement of [3H]DADLE from delta opioid receptor expressed in HEK293 cells
- ChEMBL_751948 (CHEMBL1785790) Displacement of [3H]DPDPE from delta opioid receptor in rat brain membranes
- ChEMBL_793540 (CHEMBL1932291) Displacement of [3H]DADLE from delta opioid receptor in rat cerebrum membranes
- ChEMBL_979619 (CHEMBL2421111) Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes
- ChEBML_129934 Inhibitory activity towards electrically induced contractions in mouse vas deferens expressing delta opioid receptor
- ChEBML_145496 Inhibition of [3H]naltrindole binding to human Opioid receptor delta 1 in CHO cells
- ChEBML_145634 Evaluated for inhibitory activity against Opioid receptor delta 1 of mouse vas deferens (MVD).
- ChEBML_146494 Binding affinity (in vitro) against Opioid receptor delta 1 using radio-ligand binding assay
- ChEBML_146760 Inhibition of [3H]-DPDPE binding to Opioid receptor delta 1 of rat brain membranes
- ChEBML_147148 Binding affinity was determined towards Opioid receptor delta 1 using [3H]naltrindole as radioligand
- ChEBML_147155 Compound was evaluated for binding affinity against Opioid receptor delta 1 binding assay: Inactive
- ChEBML_147162 Displacement of [3H]EK from Opioid receptor delta 1 in guinea pig brain membrane
- ChEBML_147167 Displacement of [3H]naltrindole from Opioid receptor delta 1 of guinea pig brain membranes
- ChEMBL_1277198 (CHEMBL3088918) Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells
- ChEMBL_1365294 (CHEMBL3292388) Agonist activity at delta-opioid receptor (unknown origin) by [35S]GTPgammaS binding assay
- ChEMBL_145064 (CHEMBL753995) Tested for binding activity against Opioid receptor delta 1 using [3H]DPDPE ligand
- ChEMBL_145073 (CHEMBL754004) Selective binding affinity against Opioid receptor delta 2, using [3H]DSLET as radioligand
- ChEMBL_145084 (CHEMBL753309) Tested for binding activity against Opioid receptor delta 2 using [3H]DSLET ligand
- ChEMBL_145327 (CHEMBL750415) Binding affinity towards Opioid receptor delta 1 by the displacement of [125I]-Deltorphin
- ChEMBL_145481 (CHEMBL751975) Binding affinity towards human cloned Opioid receptor delta 1 using [3H]Cl-DPDPE
- ChEMBL_145482 (CHEMBL751976) Binding affinity towards human cloned Opioid receptor delta 1 using [3H]Cl-DPDPE
- ChEMBL_145485 (CHEMBL752128) Binding affinity towards cloned human Opioid receptor delta 1 in CHO cell membranes.
- ChEMBL_145486 (CHEMBL752129) Binding affinity towards cloned human Opioid receptor delta 1 in CHO cell membranes.
- ChEMBL_145491 (CHEMBL752134) Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cells
- ChEMBL_145619 (CHEMBL753533) [3H]-Cl-DPDPE competition binding assay using human cloned opioid receptor delta 1
- ChEMBL_145901 (CHEMBL750390) Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assay
- ChEMBL_146323 (CHEMBL757532) Binding affinity for delta opioid receptor using [3H]DPDPE from mouse vas deferens
- ChEMBL_146595 (CHEMBL752699) Inhibition of [3H]- ]DSLET binding to opioid receptor delta from rat brain membrane
- ChEMBL_146767 (CHEMBL755211) Inhibition of [3H]DADLE radioligand binding to rat brain opioid receptor delta 1.
- ChEMBL_146769 (CHEMBL755213) Inhibition of radioligand [3H]DADLE binding to rat brain Opioid receptor delta 1
- ChEMBL_146890 (CHEMBL751665) Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brain
- ChEMBL_146891 (CHEMBL882036) Ability to displace [3H]DADLE from Opioid receptor delta 1 of rat brain
- ChEMBL_146918 (CHEMBL757506) Binding affinity against rat brain opioid receptor delta 1 using [3H]DPDPE radioligand
- ChEMBL_147024 (CHEMBL753665) Inhibition of [3H]- DPDPE binding to delta opioid receptor of guinea pig brain
- ChEMBL_147192 (CHEMBL759365) The binding affinity was measured using [3H]- TIPPsi against Opioid receptor delta 1
- ChEMBL_147285 (CHEMBL755438) Selective binding affinity against Opioid receptor delta 1, using [3H]DPDPE as radioligand
- ChEMBL_147317 (CHEMBL755710) Inhibition of [3H]-DADLE binding to rat brain membrane Opioid receptor delta 1
- ChEMBL_1512225 (CHEMBL3611507) Displacement of [3H]-DPDPE from human delta opioid receptor transfected in HN9.10 cells
- ChEMBL_1515760 (CHEMBL3614313) Agonist activity at delta opioid receptor in beta-funaltrexamine-treated mouse vas deferens
- ChEMBL_1552797 (CHEMBL3760690) Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells
- ChEMBL_1685447 (CHEMBL4035926) Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells
- ChEMBL_1995376 (CHEMBL4629271) Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells
- ChEMBL_223435 (CHEMBL845237) Inhibition of delta-selective antagonist binding to opioid receptor of mouse vas dferens
- ChEMBL_326600 (CHEMBL863373) Displacement of [3H]deltorphin II from delta opioid receptor in rat brain membrane
- ChEMBL_327763 (CHEMBL871133) Agonistic efficacy at human delta opioid receptor by [35S]GTP-gammaS binding assay
- ChEMBL_330098 (CHEMBL858980) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells
- ChEMBL_335164 (CHEMBL861286) Displacement of [3H]DPDPE from human delta opioid receptor expressed in HN9.10 cells
- ChEMBL_392922 (CHEMBL870416) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells
- ChEMBL_393078 (CHEMBL870429) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells
- ChEMBL_423418 (CHEMBL911093) Displacement of [3H]DPDPE from human delta opioid receptor expressed in HN9.10 cells
- ChEMBL_434305 (CHEMBL917884) Displacement of [3H]NTI from delta opioid receptor in CD1 mouse brain membranes
- ChEMBL_434330 (CHEMBL917911) Displacement of [3H]naltrindole from human opioid delta receptor expressed in CHO cells
- ChEMBL_436576 (CHEMBL904884) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO membrane
- ChEMBL_438448 (CHEMBL887548) Displacement of [3H]DPDPE from human delta opioid receptor transfected in HN9.10 cells
- ChEMBL_439346 (CHEMBL887339) Displacement of [3H]diprenorphine from delta opioid receptor expressed in human HEK293 cells
- ChEMBL_439881 (CHEMBL890202) Displacement of [125I]IOXY from human delta opioid receptor expressed in CHO cells
- ChEMBL_444081 (CHEMBL893244) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO membrane
- ChEMBL_444757 (CHEMBL895004) Displacement of [125I]IOXY from human delta opioid receptor expressed in CHO cells
- ChEMBL_465060 (CHEMBL933369) Displacement of [3H]diprenorphine from mouse delta opioid receptor expressed in HEK293 cells
- ChEMBL_469678 (CHEMBL946806) Displacement of [3H]diprenorphine from mouse delta opioid receptor expressed in CHO cells
- ChEMBL_470452 (CHEMBL932679) Displacement of [3H]diprenorphine from mouse delta opioid receptor expressed in CHO cells
- ChEMBL_471609 (CHEMBL941038) Displacement of [3H]naltrindole from human delta opioid receptor expressed in deltaC6 cells
- ChEMBL_487721 (CHEMBL1009453) Displacement of [3H]Ile5,6deltorphin-2 from delta opioid receptor in Wistar rat brain
- ChEMBL_495339 (CHEMBL1006331) Displacement of [3H]NTI from monocloned delta opioid receptor expressed in CHO cells
- ChEMBL_500504 (CHEMBL1009681) Displacement of [3H]diprenorphine from human delta opioid receptor expressed in CHO cells
- ChEMBL_500680 (CHEMBL966896) Displacement of [3H]diprenorphine from human delta opioid receptor expressed in CHO cells
- ChEMBL_515865 (CHEMBL993919) Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHOK1 cells
- ChEMBL_531191 (CHEMBL974077) Displacement of [3H]DPDPE from delta opioid receptor in ICR mouse whole brain
- ChEMBL_533285 (CHEMBL973304) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells
- ChEMBL_53570 (CHEMBL663590) inhibition of [3H]DADLE binding to delta-opioid receptor of mouse brain homogenates
- ChEMBL_540501 (CHEMBL1030605) Displacement of [3H]Naltrindole from human delta opioid receptor expressed in CHO cells
- ChEMBL_543323 (CHEMBL1022993) Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cells
- ChEMBL_558748 (CHEMBL1019877) Displacement of [3H]Naltrindole form human delta opioid receptor expressed in CHO cells
- ChEMBL_563707 (CHEMBL992671) Displacement of [3H]diprenorphine from mouse delta opioid receptor expressed in CHO cells
- ChEMBL_580496 (CHEMBL1052523) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells
- ChEMBL_583044 (CHEMBL1056543) Displacement of [3H]diprenorphine from human delta opioid receptor expressed in CHO cells
- ChEMBL_583148 (CHEMBL1062527) Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cells
- ChEMBL_590499 (CHEMBL1058546) Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptor
- ChEMBL_590504 (CHEMBL1058551) Agonist activity at human delta opioid receptor by GTP[gamma]35S binding assay
- ChEMBL_590532 (CHEMBL1059347) Displacement of [3H]DPDPE from mouse delta opioid receptor expressed in CHO cells
- ChEMBL_594976 (CHEMBL1038967) Displacement of [125I]OXY from human delta opioid receptor expressed in CHO cells
- ChEMBL_595266 (CHEMBL1043618) Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptor
- ChEMBL_596275 (CHEMBL1050691) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells
- ChEMBL_603834 (CHEMBL1045629) Displacement of [3H]DPDPE from human delta opioid receptor expressed in HN9.10 cells
- ChEMBL_615876 (CHEMBL1102710) Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain membranes
- ChEMBL_616814 (CHEMBL1099398) Displacement of [3H]DADLE from human delta opioid receptor expressed in HEK293 cells
- ChEMBL_622964 (CHEMBL1112216) Displacement of [3H]naltrindole from human delta opioid receptor expressed in deltaC6 cells
- ChEMBL_635071 (CHEMBL1119185) Displacement of [3H]DPDPE from human delta opioid receptor expressed in HEK293 cells
- ChEMBL_662059 (CHEMBL1251791) Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane
- ChEMBL_674208 (CHEMBL1274305) Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes
- ChEMBL_797688 (CHEMBL1943908) Displacement of [I125]deltorphin from delta-opioid receptor overexpressed in human HEK293 cells
- ChEMBL_967564 (CHEMBL2399074) Displacement of [3H]NTI from delta opioid receptor (unknown origin) after 1.5 hrs
- ChEMBL_146913 (CHEMBL757501) Displacement of [3H]DADLE from Opioid receptor delta 1 of rat brain membranes (DAMGO quenching mu receptor)
- ChEBML_145338 Inhibition of [125I]deltorphin binding to human delta opioid receptor from membranes of HEK293 cells
- ChEBML_146596 Inhibition of [3H]DPDPE to opioid receptor delta of rat fore brain membranes was determined
- ChEBML_146639 Compound was evaluated for its binding affinity to Opioid receptor delta 1 in rat brain
- ChEBML_147175 Inhibition of binding of [3H]-DPDPE to opioid receptor delta 1 from rat brain membrane.
- ChEBML_1685441 Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellum membrane
- ChEBML_217864 Binding affinity towards delta-opioid receptor by displacement of [3H]DADL in rat brain homogenates
- ChEBML_53589 Binding affinity against delta-opioid receptor by using [3H]DADLE as radioligand in rat brain
- ChEMBL_1348092 (CHEMBL3269121) Displacement of [3H]diprenorphine from rat delta opioid receptor expressed in rat C6 cells
- ChEMBL_1353644 (CHEMBL3271433) Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain cerebellum membrane
- ChEMBL_1353656 (CHEMBL3271445) Agonist activity at human delta opioid receptor expressed in HEK293 cells by CellKey method
- ChEMBL_1432428 (CHEMBL3385710) Displacement of [3H]DPDPE from delta opioid receptor in mouse brain membranes without cerebellum
- ChEMBL_145057 (CHEMBL753991) Binding affinity towards Opioid receptor delta 1 using [3H]- [p-CIPhe4] DPDPE as radioligand
- ChEMBL_145313 (CHEMBL751919) GTPgammaS binding in cloned human Opioid receptor delta 1 transfected into hamster ovary cells
- ChEMBL_145331 (CHEMBL750419) Binding affinity was measured against cloned human Opioid receptor delta 1 (wild-type,Wt)
- ChEMBL_1454173 (CHEMBL3363203) Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellum
- ChEMBL_145887 (CHEMBL754253) In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assay
- ChEMBL_145892 (CHEMBL754258) Inhibitory activity measured against Opioid receptor delta 1 using mouse vas deference assay (MVD).
- ChEMBL_145907 (CHEMBL750396) Opioid activity against delta-receptor of isolated mouse vas deferens(MVD) at 30 uM
- ChEMBL_146326 (CHEMBL757534) Binding affinity towards mouse delta-opioid receptor was determined using [3H]diprenorphine as radioligand
- ChEMBL_146338 (CHEMBL753787) Displacement of [3H]NLT from Opioid receptor delta 1 of adult male mouse brain.
- ChEMBL_146341 (CHEMBL753790) Inhibition of [3H]-NTI binding to Opioid receptor delta 1 from mouse brain membranes.
- ChEMBL_146610 (CHEMBL750111) Displacement of radioligand [3H]- DPDPE on Opioid receptor delta 1 in monkey brain membranes
- ChEMBL_146914 (CHEMBL757502) Binding affinity of compound evaluated for Opioid receptor delta 1 isolated from rat brain
- ChEMBL_147030 (CHEMBL753671) Inhibition of [3H]-DADLE binding to Opioid receptor delta 1 of rat brain tissue
- ChEMBL_147035 (CHEMBL753676) Binding affinity to delta-opioid receptor of rat brain using [3H]DADLE as radioligand
- ChEMBL_147062 (CHEMBL754882) In vitro binding affinity against Opioid receptor delta 1 (DPDPE) in rat brain homogenates.
- ChEMBL_147152 (CHEMBL758177) Binding affinity was determined against Opioid receptor delta 1 from guinea pig brain membranes
- ChEMBL_147172 (CHEMBL754471) Inhibition of [3H]- ]DSLET binding to Opioid receptor delta 1 from rat brain membrane
- ChEMBL_147174 (CHEMBL754473) Inhibition of [3H]-DADLE binding to Opioid receptor delta 1 of rat brain membranes
- ChEMBL_1522817 (CHEMBL3630376) Displacement of [3H]-DPDPE from delta opioid receptor (unknown origin) transfected in HEK293 cells
- ChEMBL_1552643 (CHEMBL3762582) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cell membrane
- ChEMBL_1567712 (CHEMBL3787927) Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes
- ChEMBL_1811155 (CHEMBL4310615) Displacement of [3H]-DADLE from recombinant human delta-opioid receptor expressed in HEK293 cells
- ChEMBL_181698 (CHEMBL788107) binding affinities against delta opioid receptor of rat brain using [3H]DAMGO as radioligand.
- ChEMBL_184414 (CHEMBL791516) Binding affinities against delta opioid receptor of rat brain using [3H]DAMGO as radioligand.
- ChEMBL_1923561 (CHEMBL4426517) Binding affinity to human delta opioid receptor expressed in HEK cells by PDSP assay
- ChEMBL_2164672 (CHEMBL5049533) Displacement of [3H]-DADLE from human recombinant delta opioid receptor by radioligand binding assay
- ChEMBL_223425 (CHEMBL844035) Inhibition of [3H]DPDPE binding to delta opioid receptor of guinea pig brain homogenate
- ChEMBL_223428 (CHEMBL845231) Inhibition of [3H]DPDPE binding to delta opioid receptor of guinea pig brain homogenate
- ChEMBL_303005 (CHEMBL830244) Inhibitory constant against human Opioid receptor delta 1 using [3H]diprenorphine as radio ligand
- ChEMBL_303091 (CHEMBL828763) Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain membrane
- ChEMBL_303445 (CHEMBL839705) Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranes
- ChEMBL_303454 (CHEMBL839714) Displacement of [3H[Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranes
- ChEMBL_304038 (CHEMBL840216) Binding affinity against Opioid receptor delta 1 from rat brain membranes using [3H]DADLE
- ChEMBL_325354 (CHEMBL861054) Displacement of [3H]deltorphin II from rat delta opioid receptor in brain P2 synaptosomes
- ChEMBL_326435 (CHEMBL867593) Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranes
- ChEMBL_331365 (CHEMBL867090) Displacement of [3H]naltrindole from cloned human delta opioid receptor expressed in CHO cells
- ChEMBL_364000 (CHEMBL860177) Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomes
- ChEMBL_376241 (CHEMBL869294) Inhibition of (-)-[9-3H]bremazocine binding to delta opioid receptor expressed in HEK293 cells
- ChEMBL_378703 (CHEMBL853451) Displacement of radiolabeled DPDPE-Cl from delta opioid receptor in Hartley guinea pig brain
- ChEMBL_416473 (CHEMBL907186) Displacement of [3H]diprenorphine from human recombinant delta opioid receptor expressed in C6 cells
- ChEMBL_422418 (CHEMBL909853) Displacement of [3H]diprenorphine from human cloned delta opioid receptor expressed in CHO cells
- ChEMBL_422439 (CHEMBL908255) Displacement of [3H]diprenorphine from human cloned delta opioid receptor expressed in CHO cells
- ChEMBL_423718 (CHEMBL855468) Displacement of [3H]Ile5,6-deltorphin from delta opioid receptor in Wistar rat brain membrane
- ChEMBL_424404 (CHEMBL911335) Displacement of [3H]deltorphin II from delta opioid receptor in rat synaptosomes P2 fraction
- ChEMBL_430079 (CHEMBL918101) Displacement of [3H]DPDPE from delta opioid receptor in rat brain synaptosomes P2 fraction
- ChEMBL_441143 (CHEMBL891362) Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosome
- ChEMBL_448536 (CHEMBL896540) Displacement of [3H]DPDPE from cloned delta opioid receptor expressed in CHO cell membrane
- ChEMBL_451933 (CHEMBL901091) Displacement of [3H]bremazocine from cloned human delta opioid receptor expressed in CHO cells
- ChEMBL_454477 (CHEMBL886503) Displacement of [3H]diprenorphine from human delta opioid receptor expressed in CHO cell membrane
- ChEMBL_457576 (CHEMBL922776) Activity at delta opioid receptor assessed as stimulation of [35S]GTP-gamma-S binding
- ChEMBL_471596 (CHEMBL940227) Displacement of [3H]deltorphine 2 from human delta opioid receptor expressed in CHOK1 cells
- ChEMBL_477926 (CHEMBL923551) Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cells
- ChEMBL_479226 (CHEMBL927002) Displacement of [3H]diprenorphine from human delta opioid receptor expressed in CHO-K1 cells
- ChEMBL_510226 (CHEMBL1005604) Displacement of [3H]Naltindole from human delta opioid receptor expressed in CHO cell membrane
- ChEMBL_556070 (CHEMBL953423) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cell membrane
- ChEMBL_559164 (CHEMBL1012109) Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellum
- ChEMBL_561948 (CHEMBL1021466) Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cells
- ChEMBL_572572 (CHEMBL1025188) Displacement of [3H]naltrindole from human cloned delta opioid receptor expressed in CHO cells
- ChEMBL_582245 (CHEMBL1060813) Displacement of [3H]naltrindole from human cloned delta opioid receptor expressed in CHO cells
- ChEMBL_591228 (CHEMBL1056133) Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in CHO cells
- ChEMBL_631962 (CHEMBL1104718) Displacement of [3H]deltorphine-2 from human delta opioid receptor expressed in CHOK1 cells
- ChEMBL_639786 (CHEMBL1175731) Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells
- ChEMBL_702692 (CHEMBL1657628) Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells
- ChEMBL_725831 (CHEMBL1678427) Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cells
- ChEMBL_742674 (CHEMBL1769552) Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells
- ChEMBL_772111 (CHEMBL1837877) Displacement of [3H]DPDPE from mouse delta opioid receptor in whole brain without cerebellum
- ChEMBL_814124 (CHEMBL2020765) Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellum
- ChEMBL_850392 (CHEMBL2150812) Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellum
- ChEMBL_884721 (CHEMBL2215602) Displacement of [3H]DHDPE from delta opioid receptor in mouse whole brain without cerebellum
- ChEMBL_886624 (CHEMBL2216209) Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellum
- ChEMBL_988384 (CHEMBL2437811) Displacement of [3H]DPDPE from mouse brain delta opioid receptor by scintillation counting analysis
- ChEMBL_147029 (CHEMBL753670) Binding affinity of compound was determined against Opioid receptor delta 1 from a native receptor in guinea pig
- ChEMBL_145488 (CHEMBL752131) Binding affinity towards recombinant human Opioid receptor delta 1 transfected in to CHO cells for the displacement of [3H]Cl-DPDPE (delta)
- ChEBML_147048 Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assay
- ChEMBL_145061 (CHEMBL883421) Binding affinity towards Opioid receptor delta 1 using [3H]DPDPE as radioligand in Chinese hamster ovary cells expressing cloned opioid receptors
- ChEMBL_145062 (CHEMBL753993) Binding affinity towards Opioid receptor delta 1 using [3H]DPDPE as radioligand in Chinese hamster ovary cells expressing cloned opioid receptors
- ChEBML_145186 Compound was evaluated for the agonistic activity against Opioid receptor delta 1 in hamster vas deferens.
- ChEBML_145772 Compound was evaluated for its inhibitory potency against Opioid receptor delta 1 of Mouse vas deferens
- ChEBML_145890 Inhibitory activity against Opioid receptor delta 1 of (endomorphin 2) in mouse vas deferens was determined
- ChEBML_146435 Binding affinity against opioid receptor delta from guinea pig brain membranes using [3H]DADLE as radioligand
- ChEBML_146486 Ability to induce 50% of maximal effect in mouse vas deferens expressing Opioid receptor delta 1
- ChEBML_146590 Binding affinity to opioid receptor delta was determined in rat brain using [3H]DSTBULET as radioligand
- ChEBML_146613 Binding affinity against Opioid receptor delta 1 of calf cortex using [3H]U-69593 as radioligand
- ChEBML_146874 Compound was evaluated for its inhibitory potency against Opioid receptor delta 1 of Guinea pig ileum
- ChEBML_146905 Binding affinity against delta opioid receptor by displacement of radioligand [3H]DSLET in rat brain membrane
- ChEBML_146917 Binding affinity against Opioid receptor delta 1 using [3H]DT in rat brain synaptosomes was determined
- ChEBML_147042 Binding affinity was determined as ability to displace [3H]DADLE radioligand from Opioid receptor delta 1
- ChEBML_147168 Binding affinity to Opioid receptor delta 1 using [3H]DPDPE as a radioligand in guinea pig
- ChEBML_217857 Compound was tested for its binding affinity against opioid receptor delta using [3H]DPDPE as radioligand.
- ChEMBL_1337151 (CHEMBL3240182) Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes after 2 hrs
- ChEMBL_1352785 (CHEMBL3268185) Displacement of [3H]diprenorphine from delta opioid receptor (unknown origin) expressed in CHO cells membranes
- ChEMBL_145190 (CHEMBL754435) Inhibition of [3H]naltrindole binding to opioid receptor delta 1 of Chinese hamster ovary membrane
- ChEMBL_145338 (CHEMBL750573) Inhibition of [125I]deltorphin binding to human delta opioid receptor from membranes of HEK293 cells
- ChEMBL_145467 (CHEMBL751254) Ability to displace [3H]DPDPE from human recombinant Opioid receptor delta 1 in CHO cells
- ChEMBL_145762 (CHEMBL752780) Agonist activity was evaluated in guinea pig ileum (GPI) preparations at Opioid receptor delta 1
- ChEMBL_145763 (CHEMBL752781) Agonist activity was evaluated in mouse vas deferens (MVD) preparations at Opioid receptor delta 1
- ChEMBL_145764 (CHEMBL752782) Antagonist activity against delta-opioid receptor in mouse vas deferens in the presence of DADLE
- ChEMBL_145775 (CHEMBL753431) Compound was tested for opioid receptor delta 1 agonism or antagonism in mouse vas deferens
- ChEMBL_145776 (CHEMBL753432) Compound was tested for opioid receptor delta 1 agonism or antagonism in mouse vas deferens
- ChEMBL_146342 (CHEMBL753791) Inhibitory concentration against Opioid receptor delta 1 in mouse vas deferens using competition binding assay
- ChEMBL_146343 (CHEMBL753792) Inhibitory concentration against Opioid receptor delta 1 in mouse vas deferens using competition binding assay
- ChEMBL_146430 (CHEMBL757182) Compound was evaluated for its inhibitory potency against opioid receptor delta of Guinea pig ileum
- ChEMBL_146452 (CHEMBL758727) Compound was evaluated for its inhibitory potency against opioid receptor delta of Mouse vas deferens
- ChEMBL_146639 (CHEMBL754320) Compound was evaluated for its binding affinity to Opioid receptor delta 1 in rat brain
- ChEMBL_146648 (CHEMBL754932) Inhibition of [3H][p-Cl-Phe-]DPDE binding to rat brain homogenate delta-opioid receptor
- ChEMBL_146897 (CHEMBL751671) Affinity towards human Opioid receptor delta 1 on CHO cell membranes using [3H]DPDPE displacement.
- ChEMBL_147039 (CHEMBL753342) Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomes
- ChEMBL_147064 (CHEMBL754884) Displacement of [3H]Ile5,6-deltorphin II from opioid receptor delta 1 of rat brain membranes
- ChEMBL_147137 (CHEMBL754169) Binding affinity against Delta Opioid receptor in Guinea pig brain membranes using [3H]DAMGO+DADLE
- ChEMBL_147183 (CHEMBL754482) Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.
- ChEMBL_147281 (CHEMBL755203) Inhibition of binding of [3H]DADLE to Opioid receptor delta 1 in guinea pig membranes
- ChEMBL_1504575 (CHEMBL3591316) Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assay
- ChEMBL_1552659 (CHEMBL3762758) Antagonist activity at human delta opioid receptor in CD1 mouse assessed as electrically induced twitches
- ChEMBL_1564948 (CHEMBL3783009) Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrs
- ChEMBL_166191 (CHEMBL771030) Binding affinities against delta opioid receptor of rat brain using [3H]-nor BNI as radioligand.
- ChEMBL_1672056 (CHEMBL4022085) Displacement of [3H]DPN from recombinant human delta opioid receptor expressed in CHOK1 cell membranes
- ChEMBL_1780619 (CHEMBL4252136) Displacement of [3H]DADLE from delta-opioid receptor in rat brain membranes after 2 hrs
- ChEMBL_2075854 (CHEMBL4731388) Agonist activity at human delta opioid receptor assessed as inhibition of forskolin-induced cAMP accumulation
- ChEMBL_303324 (CHEMBL840049) Inhibition of [3H]diprenorphine binding to rat Opioid receptor delta 1 expressed in C6 cells
- ChEMBL_303501 (CHEMBL839973) Inhibition of [3H]C1-DPDPE binding to human delta opioid receptor expressed in CHO cells
- ChEMBL_303535 (CHEMBL839649) Inhibition of [3H][Ile5,6]deltorphin II binding to opioid receptor delta from rat brain membranes
- ChEMBL_416465 (CHEMBL907787) Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cells
- ChEMBL_430155 (CHEMBL919064) Displacement of [3H]Cl-DPDPE from human recombinant delta opioid receptor expressed in CHO cells
- ChEMBL_439350 (CHEMBL888461) Ratio of IC50 of drug to naltrindole for delta opioid receptor in mouse vas deferens
- ChEMBL_441425 (CHEMBL891658) Binding affinity to delta opioid receptor in rat brain synaptosome membrane by radioligand binding assay
- ChEMBL_460022 (CHEMBL943141) Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cells
- ChEMBL_467788 (CHEMBL931352) Displacement of [3H]naltrindole from human cloned delta opioid receptor expressed in CHO cell membrane
- ChEMBL_482481 (CHEMBL956177) Displacement of [3H]pCl-DPDP from delta opioid receptor in rat central nervous system membrane
- ChEMBL_515869 (CHEMBL993923) Agonist activity at human delta opioid receptor expressed in CHOK1 cells by [35S]GTPgammaS binding
- ChEMBL_526494 (CHEMBL975645) Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK293 cells
- ChEMBL_540201 (CHEMBL1029830) Displacement of [3H]DPDPE from delta opioid receptor in Sprague-Dawley rat brain synaptosomal membranes
- ChEMBL_546203 (CHEMBL1036850) Displacement of [3H][Ile5,6]deltorphin-2 from delta opioid receptor in Wistar rat brain membrane
- ChEMBL_573420 (CHEMBL1061315) Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cell membrane
- ChEMBL_588102 (CHEMBL1044828) Displacement of [3H]DSLET from delta opioid receptor in rat brain by liquid scintillation counting
- ChEMBL_601075 (CHEMBL1071834) Displacement of [3H]DPDPE from delta opioid receptor expressed in HEK293 cells by visible spectrophotometry
- ChEMBL_631250 (CHEMBL1113830) Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membrane
- ChEMBL_662214 (CHEMBL1252205) Displacement of [3H]DPDPE from Sprague-Dawley rat delta opioid receptor by liquid scintillation counting
- ChEMBL_749284 (CHEMBL1785219) Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes after 2 hrs
- ChEMBL_767032 (CHEMBL1828463) Displacement of [3H]-NTI from delta opioid receptor expressed in CHO cells after 1 hr
- ChEMBL_793543 (CHEMBL1932294) Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellum
- ChEMBL_801265 (CHEMBL1947328) Displacement of radiolabeled iodinated deltorphin 2 from delta opioid receptor expressed in HEK293 cell membranes
- ChEMBL_872985 (CHEMBL2188279) Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Wistar rat brain membranes
- ChEMBL_878638 (CHEMBL2189108) Displacement of [3H]DSLET from delta opioid receptor in rat brain membranes after 2 hrs
- ChEMBL_878882 (CHEMBL2184595) Displacement of [3H]NTI from delta opioid receptor expressed in CHO cells after 1 hr
- ChEMBL_882177 (CHEMBL2215009) Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane after 2 hrs
- ChEMBL_886707 (CHEMBL2209607) Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellum
- ChEMBL_960775 (CHEMBL2387944) Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cell membranes
- ChEMBL_961552 (CHEMBL2388583) Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain devoid of cerebellum
- ChEMBL_146320 (CHEMBL757529) Binding affinity against Opioid receptor delta 1 receptor binding in ICR mouse brain membranes using the radioligand [3H]naltrindole
- ChEMBL_147288 (CHEMBL755876) The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1) antagonist
- ChEMBL_147048 (CHEMBL753275) Compound was evaluated for its binding affinity by displacement [3H]- DSLET from Opioid receptor delta 1 by using opioid radioligand binding assay
- ChEBML_129933 Inhibitory activity towards delta Opioid receptor using guinea pig ileum (GPI) assay was determined for the compound
- ChEBML_146649 Binding affinity in competition with [3H]- DPDPE in Opioid receptor delta 1 binding to rat brain membrane
- ChEBML_146763 Evaluated for the inhibition of [3H]DADLE binding to Opioid receptor delta 1 in rat brain homogenates.
- ChEBML_146866 Binding affinity against Opioid receptor delta 1 in guinea pig brain homogenate using [3H]- DPDPE as radioligand
- ChEBML_146873 Inhibition of [3H]DPDPE binding to guinea pig brain membrane Opioid receptor delta 1 at 1.0 nM
- ChEBML_146877 Inhibition of Opioid receptor delta 1 by displacing 1 nM [3H]DPDPE in guinea pig brain membrane
- ChEBML_146880 Evaluated for the inhibition of [3H]DADLE binding to Opioid receptor delta 1 of guinea pig brain
- ChEBML_146883 Inhibitory activity against Opioid receptor delta 1 of guinea pig was determined by using [3H]DADLE radioligand
- ChEBML_147017 Binding affinity against Opioid receptor delta 1 in guinea pig brain homogenates, using [3H]DPDPE as radioligand.
- ChEBML_147034 Inhibition of [3H]DPDPE radioligand binding to rat opioid receptor delta 1 site from rat brain membranes
- ChEBML_147046 Compound was evaluated for binding affinity towards Opioid receptor delta 1 by displacement of [3H]-DADLE radioligand
- ChEBML_147140 Binding affinity for delta opioid receptor was determined using radioligand [3H]DPDPE in Guinea pig brain membranes.
- ChEBML_147151 Binding affinity towards Opioid receptor delta 1 in guinea pig brain membranes using [3H]naltrindole as radioligand
- ChEBML_147292 The compound was tested for binding activity towards Opioid receptor delta 1 in guinea pig brain membranes.
- ChEBML_147330 Compound was evaluated for binding affinity towards Opioid receptor delta 1 by displacing 125 I-deltorphin II
- ChEBML_147331 In vitro binding affinity towards Opioid receptor delta 1 was determined using [3H]-DAMGO or [3H]CTOP
- ChEBML_1711445 Displacement of [3H]DADLE from human recombinant delta opioid receptor after 60 mins by scintillation counting analysis
- ChEBML_217729 Binding affinity towards delta opioid receptor in guinea pig brain membranes using [3H]- CI-DPDPE as radioligand
- ChEBML_53588 Binding affinity evaluated by inhibition of binding of [3H]DADLE to delta opioid receptor of rat brain
- ChEMBL_1275491 (CHEMBL3090461) Displacement of [3H]-naltrindole from human delta opioid receptor transfected in CHO cells after 3 hrs
- ChEMBL_1277323 (CHEMBL3089284) Agonist activity at human delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assay
- ChEMBL_1339025 (CHEMBL3243891) Displacement of [3H]-diprenorphine from human delta opioid receptor after 120 mins by cell based assay
- ChEMBL_1363047 (CHEMBL3293116) Binding affinity to human cloned delta opioid receptor expressed in CHO cells by radioligand displacement assay
- ChEMBL_1433275 (CHEMBL3388813) Agonist activity at human delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assay
- ChEMBL_1437486 (CHEMBL3387857) Agonist activity at mouse delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assay
- ChEMBL_145322 (CHEMBL750410) Binding affinity against human opioid receptor delta 1 using [125I]-[D-Ala2]-deltorphin II as radioligand
- ChEMBL_145336 (CHEMBL750571) In vitro binding affinity against cloned human Opioid receptor delta 1 expressed in HEK 293S cells
- ChEMBL_145466 (CHEMBL751253) Displacement of [3H]C1-DPDPE from human recombinant Opioid receptor delta 1 on CHO cell membranes.
- ChEMBL_145492 (CHEMBL872958) Competitive binding displacement analyses was performed from permanently transfected HEK293 cells expressing Opioid receptor delta 1
- ChEMBL_1455711 (CHEMBL3366386) Displacement of [3H]diprenorphine from human delta opioid receptor expressed in HEK293 cells by scintillation counting
- ChEMBL_145772 (CHEMBL753428) Compound was evaluated for its inhibitory potency against Opioid receptor delta 1 of Mouse vas deferens
- ChEMBL_145890 (CHEMBL754256) Inhibitory activity against Opioid receptor delta 1 of (endomorphin 2) in mouse vas deferens was determined
- ChEMBL_145895 (CHEMBL754260) Inhibitory concentration against delta opioid receptor of electrically induced smooth muscle contraction of mouse vas deferens
- ChEMBL_146037 (CHEMBL754944) Binding assay evaluated using DPPE radioligand in CHO cells transfected with mouse Opioid receptor delta 1
- ChEMBL_1461562 (CHEMBL3396803) Agonist activity at human delta opioid receptor expressed in COS7 cells after 60 mins IP1 assay
- ChEMBL_146318 (CHEMBL758108) Antagonist activity of compound on agonist stimulated [35S]GTP-gamma-S binding on delta-opioid receptor
- ChEMBL_146321 (CHEMBL757530) Binding affinity against Opioid receptor delta 1 using [3H][D-Ala2, D-Leu5]-enkephalin as radioligand
- ChEMBL_146591 (CHEMBL750213) Inhibition of [3H]-DADLE binding to opioid receptor delta in P2 membrane preparation of rat brain
- ChEMBL_146599 (CHEMBL752703) The compound was tested for the ability to displace opioid receptor delta specific radioligand [3H]-DSLET
- ChEMBL_146613 (CHEMBL750114) Binding affinity against Opioid receptor delta 1 of calf cortex using [3H]U-69593 as radioligand
- ChEMBL_146652 (CHEMBL754936) Binding affinity was measured against Opioid receptor delta 1 using [3H]p-Cl-DPDPE as radioligand.
- ChEMBL_146755 (CHEMBL753335) Compound was evaluated for its inhibitory potency against Opioid receptor delta 1 of Mouse vas deferens
- ChEMBL_146766 (CHEMBL755210) In vitro inhibition of [3H]deltorphin binding to Opioid receptor delta 1 using rat brain membranes.
- ChEMBL_146901 (CHEMBL751114) Binding activity against Opioid receptor delta 1 using [3H]DADLE as radioligand in rat brain membranes.
- ChEMBL_146904 (CHEMBL751117) Binding affinity against Opioid receptor delta 1 of rat brain using [3H]-nor BNI as radioligand.
- ChEMBL_146905 (CHEMBL751118) Binding affinity against delta opioid receptor by displacement of radioligand [3H]DSLET in rat brain membrane
- ChEMBL_146906 (CHEMBL751119) Binding affinity at opioid receptor delta 1 by displacement of [3H]DADLE in rat brain membrane
- ChEMBL_146920 (CHEMBL757508) Binding affinity for Opioid receptor delta 1 using [3H]DPDPE in rat brain P2 synaptosomal preparation
- ChEMBL_146922 (CHEMBL757314) Binding affinity on HEK293 cells transiently transfected with plasmids encoding the rat Opioid receptor delta 1
- ChEMBL_147010 (CHEMBL756213) Ability to inhibit GTP-gamma-S binding to Opioid receptor delta 1 of guinea pig caudate
- ChEMBL_147011 (CHEMBL756214) Ability to inhibit GTP-gamma-S binding to Opioid receptor delta 1 of guinea pig caudate.
- ChEMBL_147019 (CHEMBL756221) Binding affinity against Opioid receptor delta 1 in guinea pig brain membranes using [3H]Cl-DPDPE
- ChEMBL_147020 (CHEMBL756222) Binding affinity against Opioid receptor delta 1 using [3H]DADLE as radioligand in guinea pig brain
- ChEMBL_147022 (CHEMBL753663) Binding affinity against Opioid receptor delta 1 in guinea pig brain membranes using [3H]Cl-DPDPE
- ChEMBL_147038 (CHEMBL753341) Binding affinity towards Opioid receptor delta 1 using [3H]CI-DPDPE as radioligand in rat brain
- ChEMBL_147143 (CHEMBL754175) Binding affinity to displace radioligand [3H]naltrindole on Opioid receptor delta 1 in guinea pig membranes.
- ChEMBL_147150 (CHEMBL758175) Binding affinity towards Opioid receptor delta 1 from guinea pig brain using [3H]naltrindole as radioligand
- ChEMBL_147157 (CHEMBL758768) Compound was evaluated for binding affinity at Opioid receptor delta 1 in guinea pig brain membranes
- ChEMBL_147193 (CHEMBL756869) The binding affinity was measured using [3H]-DIDII against Opioid receptor delta 1 of rat brain
- ChEMBL_147194 (CHEMBL756870) The binding affinity was measured using [3H]naltrindole against Opioid receptor delta 1 of rat brain
- ChEMBL_1512228 (CHEMBL3611510) Agonist activity at human delta opioid receptor transfected in HN9.10 cells by [35S]GTPgammaS binding assay
- ChEMBL_1521809 (CHEMBL3626669) Displacement of [3H]diprenorphine from FLAG-tagged mouse delta opioid receptor expressed in CHO cell membranes
- ChEMBL_1548299 (CHEMBL3755750) Displacement of [3H]DPDPE from human delta opioid receptor after 180 mins by scintillation counting analysis
- ChEMBL_1552649 (CHEMBL3762588) Partial agonist activity at delta opioid receptor (unknown origin) assessed as inhibition of adenylyl cyclase activity
- ChEMBL_1552653 (CHEMBL3762592) Agonist activity at rat delta opioid receptor transfected in C6 cells by [35S]GTPgammaS binding assay
- ChEMBL_1552798 (CHEMBL3760691) Agonist activity at human delta-opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assay
- ChEMBL_1906989 (CHEMBL4409347) Inhibition of delta opioid receptor (unknown origin) in presence of DAMGO by [35S]-GTPgammaS binding assay
- ChEMBL_1906991 (CHEMBL4409349) Inhibition of delta opioid receptor (unknown origin) in presence of DPDPE by [35S]-GTPgammaS binding assay
- ChEMBL_217732 (CHEMBL823796) Binding affinity towards human delta opioid receptor in CHO cells using [3H]- CI-DPDPE as radioligand
- ChEMBL_217857 (CHEMBL822180) Compound was tested for its binding affinity against opioid receptor delta using [3H]DPDPE as radioligand.
- ChEMBL_303256 (CHEMBL826382) Binding affinity against Opioid receptor delta 1 expressed in CHO cells using [3H]Naltrindole as radioligand
- ChEMBL_306417 (CHEMBL828088) In vitro inhibitory concentration against Opioid receptor delta 1 was measured using mouse vas deferens assay
- ChEMBL_321479 (CHEMBL880420) Binding affinity against human opioid receptor delta 1 expressed in HEK293 cells using [3H]DDPDE radioligand
- ChEMBL_335168 (CHEMBL861290) Inhibition of [35S]GTP-gamma-S binding to human delta opioid receptor expressed in CHO cells
- ChEMBL_392088 (CHEMBL871071) Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane
- ChEMBL_424406 (CHEMBL911337) Activity at delta opioid receptor assessed as inhibition of muscle contraction in mouse vas deferens assay
- ChEMBL_434265 (CHEMBL918425) Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membrane
- ChEMBL_434962 (CHEMBL919363) Displacement of [125I]deltorphin 2 from human recombinant delta opioid receptor expressed in HEK cell membranes
- ChEMBL_448540 (CHEMBL897689) Agonist activity at human delta opioid receptor expressed in CHO membrane by [35S]GTPgammaS binding assay
- ChEMBL_457105 (CHEMBL924481) Displacement of [3H]p-Cl-DPDPE from rat recombinant delta opioid receptor expressed in C6 cells
- ChEMBL_460086 (CHEMBL924962) Displacement of [3H]deltorphin 2 from delta opioid receptor in Wistar rat brain after 45 mins
- ChEMBL_470715 (CHEMBL934556) Agonist activity at delta opioid receptor assessed as inhibition of electrically-stimulated mouse vas deferens contraction
- ChEMBL_473938 (CHEMBL950318) Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane
- ChEMBL_510432 (CHEMBL1003108) Displacement of [3H]deltorphin2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane
- ChEMBL_53450 (CHEMBL666300) Agonistic activity towards Opioid receptor delta 1 as inhibitory activity towards electrically stimulated mouse vas deferens
- ChEMBL_577730 (CHEMBL1063990) Displacement of [3H]DPDE from delta opioid receptor in rat brain membrane by liquid scintillation counting
- ChEMBL_580505 (CHEMBL1053219) Displacement of [3H]p-Cl-DPDPE from rat delta opioid receptor expressed in rat C6 cells
- ChEMBL_588903 (CHEMBL1061227) Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]GTPgammaS binding
- ChEMBL_591866 (CHEMBL1045070) Agonist activity at delta opioid receptor in mouse vas deferens assessed as effect on muscle contraction
- ChEMBL_601081 (CHEMBL1071840) Activity at delta opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS binding
- ChEMBL_664323 (CHEMBL1259358) Antagonist activity at human delta opioid receptor assessed as inhibition of SNC80-stimulated [35S]GTPgammaS binding
- ChEMBL_750583 (CHEMBL1786447) Displacement of [3H]DPN from human recombinant delta-type opioid receptor expressed in CHO cell membranes
- ChEMBL_856832 (CHEMBL2163097) Agonist activity at delta opioid receptor expressed in CHO-hg cells by [35S]-GTPgammaS binding assay
- ChEMBL_957479 (CHEMBL2378217) Displacement of [3H]-enkephalin from human delta opioid receptor transfected in CHOK1 cells after 60 mins
- ChEMBL_980540 (CHEMBL2422699) Displacement of [3H]-naltrindole from mouse delta opioid receptor expressed in CHO cells after 1.5 hrs
- ChEBML_147165 Compound was tested for the inhibition of [35S]GTP-gamma-S, binding in Guinea pig Caudate stimulated by the Opioid receptor delta 1 agonist Delta-SNC80
- ChEBML_145479 Binding affinity for human opioid receptor delta 1 using [3H]- CL-DPDPE as radioligand transfected into CHO cells
- ChEBML_146446 Tested for inhibitory effect on binding of [3H]DPDPE to opioid receptor delta in guinea pig cerebellum membranes
- ChEBML_147051 Binding affinity against Opioid receptor delta 1 in P2 membrane preparation of rat brain by [3H]DADLE displacement.
- ChEBML_147139 Binding affinity against Opioid receptor delta 1 was determined in brain membrane preparations from male Hartley guinea-pigs
- ChEBML_147186 Tested for binding affinity against delta opioid receptor by displacing [3H]- DSLET radioligand from rat brain membrane preparations
- ChEBML_147344 Tested for binding affinity towards Opioid receptor delta 1 in rat and guinea pig brain membrane binding assays
- ChEMBL_1335003 (CHEMBL3239390) Displacement of [3H]deltorphin-2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membranes
- ChEMBL_1353650 (CHEMBL3271439) Agonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]-GTP[gammaS] binding
- ChEMBL_1367237 Displacement of [3H]-deltorphin 2 from human delta-opioid receptor transfected in CHO-K1 cell by scintillation counting
- ChEMBL_145183 (CHEMBL754283) Binding affinity for Opioid receptor delta 1 as inhibition of [3H]DADAL binding to rat brain membranes
- ChEMBL_145334 (CHEMBL750422) Binding inhibition of [3H]- -naltrindole (0.15 nM) to membranes in CHO cells expressing Opioid receptor delta 1
- ChEMBL_145471 (CHEMBL751258) Binding affinity against cloned human Opioid receptor delta 1 transfected onto CHO cells using [3H]Cl-DPDPE
- ChEMBL_145493 (CHEMBL752135) Competitive binding displacement analyses was performed from permanently transfected HEK293 cells expressing human Opioid receptor delta 1
- ChEMBL_145770 (CHEMBL752788) Compound is tested in vitro in mouse vas deferens (MVD) assay mediated by Opioid receptor delta 1
- ChEMBL_145778 (CHEMBL755220) Functional biological activity for Opioid receptor delta 1 was determined in vitro, on mouse vas deferens (MVD).
- ChEMBL_145779 (CHEMBL883396) In vitro agonist activity for Opioid receptor delta 1 was determined in a mouse vas deferens assay
- ChEMBL_1462886 (CHEMBL3399798) Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in HEK cells after 60 mins
- ChEMBL_146317 (CHEMBL758864) Antagonist activity of compound on SNC 80 stimulated [35S]GTP-gamma-S binding to delta-opioid receptor
- ChEMBL_146330 (CHEMBL757538) Compound was evaluated for binding affinity against delta opioid receptor of mouse vas deferens using [3H]-DPDPE
- ChEMBL_146344 (CHEMBL753793) Ki value determined against Opioid receptor delta 1 using [3H]DPDPE at the Kd concentration 2.1 nM
- ChEMBL_146345 (CHEMBL753794) The compound tested for agonistic activity against Opioid receptor delta 1 using [3H]- NT1 as the radioligand.
- ChEMBL_146582 (CHEMBL754816) Compound was evaluated for the binding affinity in comparison with [3H]- DPDPE (opioid receptor delta selective ligand)
- ChEMBL_146641 (CHEMBL754925) The binding affinity was evaluated against [3H]dalamid binding to rat brain membranes (Opioid receptor delta 1)
- ChEMBL_146649 (CHEMBL754933) Binding affinity in competition with [3H]- DPDPE in Opioid receptor delta 1 binding to rat brain membrane
- ChEMBL_146754 (CHEMBL753334) Inhibitory activity against forskolin-stimulated cAMP production in chinese hamster ovary cells expressing Opioid receptor delta 1
- ChEMBL_146758 (CHEMBL753486) Compound was evaluated for the binding affinity in comparison with [3H]- DPDPE (delta opioid receptor selective ligand)
- ChEMBL_146883 (CHEMBL751658) Inhibitory activity against Opioid receptor delta 1 of guinea pig was determined by using [3H]DADLE radioligand
- ChEMBL_146894 (CHEMBL751668) Ability to inhibit the binding of [3H]DSLET to Opioid receptor delta 1 in rat brain membranes
- ChEMBL_146903 (CHEMBL751116) Binding affinity against Opioid receptor delta 1 by displacement of radioligand [3H]DSLET in rat brain membrane
- ChEMBL_146997 (CHEMBL753818) Tested for the binding affinity against the Delta opioid receptor in guinea pig brain using [3H]DPDPE
- ChEMBL_147025 (CHEMBL753666) Binding affinity against opioid receptor delta 1 using [3H]naltrindole as radioligand in guinea pig brain membranes.
- ChEMBL_147026 (CHEMBL753667) Binding affinity determined on Opioid receptor delta 1 in Guinea pig brain membranes using radioligand [3H]DADLE
- ChEMBL_147034 (CHEMBL753675) Inhibition of [3H]DPDPE radioligand binding to rat opioid receptor delta 1 site from rat brain membranes
- ChEMBL_147052 (CHEMBL753279) Compound was tested for binding affinity towards delta-opioid receptor in rat forebrain membrane using [3H]DPDPE
- ChEMBL_147151 (CHEMBL758176) Binding affinity towards Opioid receptor delta 1 in guinea pig brain membranes using [3H]naltrindole as radioligand
- ChEMBL_147178 (CHEMBL754477) Inhibitory activity against Opioid receptor delta 1 in rat brain membranes using [3H]DADLE as a radioligand.
- ChEMBL_147345 (CHEMBL873918) The compound tested for agonistic activity against Opioid receptor delta 1 using [3H]- NT1 as the radioligand.
- ChEMBL_1511478 (CHEMBL3606827) Displacement of [3H]DPDPE from delta opioid receptor in mouse brain membranes by liquid scintillation counting method
- ChEMBL_1552636 (CHEMBL3762575) Displacement of [3H]DPN from human delta opioid receptor expressed in CHO cells by liquid scintillation counting
- ChEMBL_1567710 (CHEMBL3787925) Agonist activity at human delta opioid receptor expressed in CHO cell membranes by [35S]GTPgammaS binding assay
- ChEMBL_1588475 (CHEMBL3826758) Displacement of [3H]DSLET from delta-type opioid receptor in rat brain membranes incubated for 2 hrs
- ChEMBL_1620923 (CHEMBL3863206) Activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_1714219 (CHEMBL4124268) Agonist activity at delta-opioid receptor in mouse vasa deferens assessed as inhibition of electrically induced contractions
- ChEMBL_1721391 (CHEMBL4136391) Displacement of [3H][Ile5,6]-deltorphin II from delta-type opioid receptor in Sprague-Dawley rat brain membranes
- ChEMBL_1780609 (CHEMBL4252126) Antagonist activity at human delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS
- ChEMBL_1906941 (CHEMBL4409299) Inhibition of full length delta opioid receptor (unknown origin) assessed as increase in beta arrestin 1 recruitment
- ChEMBL_1906942 (CHEMBL4409300) Inhibition of full length delta opioid receptor (unknown origin) assessed as increase in beta arrestin 2 recruitment
- ChEMBL_1906964 (CHEMBL4409322) Inhibition of delta opioid receptor (unknown origin) expressed in human UO5S cells by [35S]-GTPgammaS binding assay
- ChEMBL_1995381 (CHEMBL4629276) Agonist activity at human delta opioid receptor expressed in CHO cell membranes by [35S]GTPgammaS binding assay
- ChEMBL_2164690 (CHEMBL5049551) Antagonist activity at human recombinant delta opioid receptor assessed as reduction in SNC80 induced [3S]-GTPgammaS binding
- ChEMBL_217727 (CHEMBL823791) Binding affinities against delta 2 opioid receptor of rat brain using [3H]Ile5,6-deltorphin II as radioligand.
- ChEMBL_217866 (CHEMBL822189) Binding affinities against delta 2 opioid receptor of rat brain using [3H]Ile5,6-deltorphin II as radioligand.
- ChEMBL_349388 (CHEMBL865695) Activity against delta opioid receptor by stimulation of [35S]GTP-gamma-S binding in CHO-hgamma cells
- ChEMBL_392092 (CHEMBL869898) Agonist activity at delta opioid receptor assessed as inhibition of electrically-evoked contraction of mouse vas deferens
- ChEMBL_423420 (CHEMBL911095) Activity at human delta opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assay
- ChEMBL_430082 (CHEMBL917185) Agonistic activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked twitch
- ChEMBL_436683 (CHEMBL904992) Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosome membrane
- ChEMBL_441428 (CHEMBL891653) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-induced twitches
- ChEMBL_443019 (CHEMBL892151) Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane
- ChEMBL_449775 (CHEMBL898880) Displacement of [3H]deltorphin 2 from delta-opioid receptor in Sprague-Dawley rat brain P2 synaptosome membrane
- ChEMBL_455044 (CHEMBL887073) Agonist activity at human cloned delta opioid receptor assessed as stimulation of [35S]GTP-gamma-S binding
- ChEMBL_473941 (CHEMBL950321) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked-contraction
- ChEMBL_53438 (CHEMBL666288) Binding to delta opioid receptor by using [3H]DPDPE as radioligand in guinea pig brain minus cerebellum
- ChEMBL_534603 (CHEMBL989028) Agonist activity at human delta opioid receptor in CHO cells assessed as stimulation of [35S]GTPgammaS binding
- ChEMBL_534707 (CHEMBL982796) Antagonist activity against delta opioid receptor in mouse vas deference assessed as effect on DPDPE-induced response
- ChEMBL_53588 (CHEMBL665476) Binding affinity evaluated by inhibition of binding of [3H]DADLE to delta opioid receptor of rat brain
- ChEMBL_539198 (CHEMBL1024702) Agonist activity at human delta opioid receptor expressed in mouse HN9.10 cells by [35S]GTPgammaS binding assay
- ChEMBL_556073 (CHEMBL953426) Agonist activity at human delta opioid receptor expressed in CHO cell membrane by [35S]GTPgammaS binding assay
- ChEMBL_556846 (CHEMBL964706) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated contraction
- ChEMBL_575383 (CHEMBL1027057) Agonist activity at human recombinant delta opioid receptor expressed in HEK293 cells by [35S]GTPgammaS binding assay
- ChEMBL_575384 (CHEMBL1027058) Agonist activity at human recombinant delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assay
- ChEMBL_577733 (CHEMBL1052368) Agonist activity at delta opioid receptor in mouse vas deference assessed as inhibition of electrically-stimulated contraction
- ChEMBL_582956 (CHEMBL1055012) Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane
- ChEMBL_582960 (CHEMBL1055016) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contraction
- ChEMBL_586039 (CHEMBL1063596) Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by liquid scintillation counting
- ChEMBL_601677 (CHEMBL1049575) Displacement of [3H]bremazocine from mouse delta opioid receptor expressed in HEK293 cells by liquid scintillation counting
- ChEMBL_603843 (CHEMBL1046460) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated contraction
- ChEMBL_607037 (CHEMBL1074665) Displacement of [125I]diprenorphine from human delta opioid receptor expressed in CHO cells by liquid scintillation counting
- ChEMBL_630234 (CHEMBL1105636) Displacement of [3H]deltorphin-2 from delta opioid receptor from Wistar rat brain by liquid scintillation counting
- ChEMBL_633487 (CHEMBL1119299) Agonist activity at human recombinant delta opioid receptor expressed in CHO cells by [35S]GTPgammaS binding assay
- ChEMBL_635069 (CHEMBL1119183) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contraction
- ChEMBL_647233 (CHEMBL1217374) Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membrane
- ChEMBL_647573 (CHEMBL1217620) Agonist activity at human opioid delta receptor expressed in mouse HN9.10 cells assessed as [35S]GTPgammaS binding
- ChEMBL_742683 (CHEMBL1769561) Agonist activity at human opioid delta receptor expressed in mouse HN9.10 cells assessed as [35S]GTPgammaS binding
- ChEMBL_771172 (CHEMBL1837089) Displacement of [3H]Ile-deltorphin-2 from rat brain delta-type opioid receptor by liquid scintillation counting
- ChEMBL_876451 (CHEMBL2187203) Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells by scintillation counting analysis
- ChEMBL_960774 (CHEMBL2387943) Inhibition of delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_987441 (CHEMBL2438615) Displacement of [125I]-BNtxA from mouse cloned delta opioid receptor expressed in CHO cells after 90 mins
- ChEBML_145494 Compound was evaluated for functional opioid activity by stimulation of [35S]GTP-gamma-S, in cloned human Opioid receptor delta 1 transfected into CHO cells
- ChEMBL_145838 (CHEMBL755496) Displacement of [3H]dynorphin A from Opioid receptor kappa 1 of rat brain membranes (DAMGO/DADLE quenching of mu/delta receptor binding)
- ChEMBL_145494 (CHEMBL752136) Compound was evaluated for functional opioid activity by stimulation of [35S]GTP-gamma-S, in cloned human Opioid receptor delta 1 transfected into CHO cells
- ChEBML_145777 Concentration required for 50% inhibition of electrically induced contraction of the mouse vas deferens mediated through delta opioid receptor
- ChEBML_146616 Compound was tested for Inhibition of 9 (1 nM) binding to Opioid receptor delta 1 from bovine striatal Membranes
- ChEBML_146646 Ability to displace [3H]DPDPE from Opioid receptor delta 1 in rat brain membranes, was determined from radioreceptor assay.
- ChEBML_146761 Evaluated for its affinity towards Opioid receptor delta 1 in rat fore brain by displacing the radioligand [3H]DPDPE.
- ChEBML_147044 Binding affinity was determined towards Opioid receptor delta 1 in rat brain synaptosomes using [3H]deltorphin II as radioligand.
- ChEBML_147145 Binding affinity towards Opioid receptor delta 1 was determined using [d-Ser2, Leu5, Thr6] enkephalin (DSLET) as the radioligand.
- ChEBML_1651359 Displacement of [3H]DPDPE from delta opioid receptor in Sprague-Dawley rat brain membranes by liquid scintillation counter method
- ChEBML_1688146 Displacement of [3H]DADLE from delta opioid receptor in rat brain after 60 mins by liquid scintillation counting method
- ChEBML_1693459 Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by microbeta scintillation counting analysis
- ChEMBL_1277416 (CHEMBL3089527) Displacement of [3H]NTI from delta opioid receptor (unknown origin) expressed in CHO cell membranes after 1.5 hrs
- ChEMBL_1335007 (CHEMBL3239394) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_1337157 (CHEMBL3240188) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_1352796 (CHEMBL3268196) Inhibition of delta opioid receptor (unknown origin) using SNC-80 by high content imaging beta-arrestin translocation assay
- ChEMBL_1447932 (CHEMBL3379235) Displacement of [3H]-deltorphine from human delta opioid receptor expressed in CHO-K1 cells by scintillation counting analysis
- ChEMBL_145316 (CHEMBL751922) Stimulation of [35S]GTP-gamma-S, binding at human recombinant Opioid receptor delta 1 transfected into CHO cells.
- ChEMBL_145335 (CHEMBL750570) Inhibition of binding of [3H]- -naltrindole (0.15 nM) to membranes from CHO cells expressing Opioid receptor delta 1
- ChEMBL_145337 (CHEMBL750572) Inhibition of [3H][D-Ala2,D-Leu5]enkephalin binding to human Opioid receptor delta 1 in CHO cells
- ChEMBL_1454175 (CHEMBL3363205) Agonist activity at human delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]-GTPgammaS binding
- ChEMBL_145472 (CHEMBL751259) Binding affinity against human opioid receptor delta 1 transfected on CHO cells was determined using [3H]Cl-DPDPE
- ChEMBL_145608 (CHEMBL749751) Inhibition of [3H]naltrindole (0.55 nM) binding from human Opioid receptor delta 1 expressed in CHO-K1 cells.
- ChEMBL_1456849 (CHEMBL3367582) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_145768 (CHEMBL752786) Binding affinity towards Opioid receptor delta 1 by the displacement of [3H]deltorphin-II in mouse spinal cord
- ChEMBL_146316 (CHEMBL758863) In vitro binding affinity to human Opioid receptor delta 1 on CHO cell membranes using [3H]diprenorphine displacement.
- ChEMBL_146770 (CHEMBL857690) Inhibition of binding of radioligand [3H][p-Cl-phe]-DPDPE to Opioid receptor delta 1 in rat brain
- ChEMBL_146771 (CHEMBL755214) Inhibitory activity measured against [3H]DPDPE (Opioid receptor delta 1 ligand) in rat brain using radioreceptor binding assays.
- ChEMBL_146772 (CHEMBL755215) Inhibitory concentration was evaluated against delta opioid receptor by the displacement of tritiated DSLET from rat brain membranes
- ChEMBL_146868 (CHEMBL752611) Binding affinity for delta opioid receptor in guinea pig brain membranes, using 2 nM [3H]DPDPE as radioligand
- ChEMBL_146869 (CHEMBL749997) Binding affinity for delta opioid receptor in guinea pig brain membranes; using 2 nM [3H]DPDPE as radioligand
- ChEMBL_1468974 (CHEMBL3412631) Displacement of [3H]DPDPE from rat cortex delta opioid receptor after 2.5 hrs by liquid scintillation counting analysis
- ChEMBL_146898 (CHEMBL751672) Affinity was assessed using competitive binding assay labeled with [3H]DPDPE (6.3 nM) for Opioid receptor delta 1
- ChEMBL_146899 (CHEMBL751673) Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement.
- ChEMBL_146902 (CHEMBL751115) Binding affinities against Opioid receptor delta 1 of rat brain using [3H]p-Cl-Phe4-DPDPE as radioligand.
- ChEMBL_146907 (CHEMBL751120) Binding affinity for Opioid receptor delta 1 determined by displacing [3H]-DSLET from rat brain membrane binding sites
- ChEMBL_146909 (CHEMBL757497) Binding affinity measured against [3H]DPDPE (Opioid receptor delta 1 ligand) in rat brain using radioreceptor binding assays.
- ChEMBL_146910 (CHEMBL757498) Binding affinity towards human Opioid receptor delta 1 on NxG108CC15 (human neuroglioblastoma) cell membranes by [3H]DPDPE displacement.
- ChEMBL_146924 (CHEMBL757316) Binding affinity towards Opioid receptor delta 1 by the displacement of [3H]DADLE radioligand in rat brain membranes
- ChEMBL_147033 (CHEMBL753674) Binding affinity determined by displacing [3H][Ile5,6]deltorphin II from opioid receptor delta 1 in rat brain membranes
- ChEMBL_147149 (CHEMBL758174) Binding affinity towards Opioid receptor delta 1 by displacing the radioligand [3H]naltrindole from guinea pig brain membrane
- ChEMBL_147186 (CHEMBL754485) Tested for binding affinity against delta opioid receptor by displacing [3H]- DSLET radioligand from rat brain membrane preparations
- ChEMBL_147279 (CHEMBL755201) Inhibition of [35S]GTP-gamma-S, binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1)
- ChEMBL_147303 (CHEMBL857861) Binding affinity using guinea pig brain membrane preparations, towards Opioid receptor delta 1 using [3H]DPDPE as radioligand
- ChEMBL_1501217 (CHEMBL3587785) Displacement of [3H]DPDPE from delta opioid receptor (unknown origin) transfected into HEK293 cells by microplate scintillation counting
- ChEMBL_1512230 (CHEMBL3611626) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_1515752 (CHEMBL3614305) Displacement of [3H]-DPDPE from human delta opioid receptor transfected in HN9.10 cell membranes by scintillation counting analysis
- ChEMBL_1517225 (CHEMBL3620209) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated muscle contraction
- ChEMBL_1525034 (CHEMBL3637632) Displacement of [3H]-DPDPE from delta opioid receptor in rat brain membrane after 120 mins by scintillation counting
- ChEMBL_1549025 (CHEMBL3756644) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electric stimulation-induced contraction
- ChEMBL_1552648 (CHEMBL3762587) Partial agonist activity at delta opioid receptor (unknown origin) assessed as [35S]GTPgammaS binding by cell based assay
- ChEMBL_1552652 (CHEMBL3762591) Displacement of [3H]diprenorphine from rat delta opioid receptor transfected in C6 cells by liquid scintillation counting assay
- ChEMBL_1564946 (CHEMBL3783007) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_1721380 (CHEMBL4136380) Agonist activity at delta-type opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated contractions
- ChEMBL_177587 (CHEMBL783508) Inhibitory concentration was evaluated against delta opioid receptor by the displacement of tritiated DSLET from rat brain membranes
- ChEMBL_1884534 (CHEMBL4386116) Displacement of [3H]DPDPE from delta opioid receptor in rat membranes after 120 mins by scintillation counting analysis
- ChEMBL_1906940 (CHEMBL4409298) Inhibition of full length delta opioid receptor (unknown origin) assessed as inhibition of forskolin-stimulated intracellular cAMP accumulation
- ChEMBL_1995388 (CHEMBL4629283) Inverse agonist activity at human delta opioid receptor expressed in CHO cell membranes by [35S]GTPgammaS binding assay
- ChEMBL_2106124 (CHEMBL4814799) Displacement of [3H]-DPDPE from human delta opioid receptor expressed in CHO-K1 cells by radioligand binding assay
- ChEMBL_2169948 (CHEMBL5055007) Displacement of [3H]-DPDPE from human delta opioid receptor expressed in mouse HN9.10 cells by radioligand binding assay
- ChEMBL_2494529 Displacement of [3H]DPDPE from human cloned delta-opioid receptor expressed in CHO cell membrane by liquid scintillation counting
- ChEMBL_304325 (CHEMBL829297) Stimulation of [35S]-GTP gammaS binding to Opioid receptor delta 1 expressed in CHO cells; ND = Not determined
- ChEMBL_335170 (CHEMBL861292) Agonist activity at delta opioid receptor by inhibition of muscle contraction in electrically stimulated isolated mouse vas deferens
- ChEMBL_425710 (CHEMBL913692) Agonist activity at delta opioid receptor by inhibition of electrically evoked muscle contraction in isolated mouse vas deferens
- ChEMBL_430160 (CHEMBL919069) Activity at human recombinant delta opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assay
- ChEMBL_436688 (CHEMBL904997) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_441147 (CHEMBL891366) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractions
- ChEMBL_449059 (CHEMBL899317) Antagonist activity at human delta opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assay
- ChEMBL_449630 (CHEMBL898725) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_491468 (CHEMBL949524) Displacement of [3H][D-Ala2,D-Leu5]enkephalin from human cloned delta opioid receptor expressed in CHO cells
- ChEMBL_510435 (CHEMBL1003111) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_53593 (CHEMBL665481) Effective concentration for agonistic activity towards delta opioid receptor was determined by [35S]GTP-gamma-S functional assay
- ChEMBL_543332 (CHEMBL1023002) Agonist activity at human delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding
- ChEMBL_565187 (CHEMBL958393) Agonist activity at human delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding
- ChEMBL_573426 (CHEMBL1061321) Agonist activity at human delta opioid receptor expressed in mouse HN9.10 cell membrane by [35S]GTPgamma binding assay
- ChEMBL_573491 (CHEMBL1063044) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_578688 (CHEMBL1063069) Displacement of [3H]diprenorphine from human delta opioid receptor expressed in CHO cells by Topcount microplate scintillation counting
- ChEMBL_583045 (CHEMBL1056544) Agonist activity at human delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding
- ChEMBL_588897 (CHEMBL1061221) Displacement of [3H]DPDPE from human recombinant delta opioid receptor expressed in CHO cells by liquid scintillation counting
- ChEMBL_591213 (CHEMBL1058519) Displacement of [3H]DPDPE from delta opioid receptor expressed in CHO cells after 90 mins by scintillation counting
- ChEMBL_591224 (CHEMBL1059302) Inhibition of radiolabeled [D-Ala2,MePhe4,Gly-ol5]enkephalin binding to delta opioid receptor in rat brain membrane
- ChEMBL_601119 (CHEMBL1074534) Inverse agonist activity at delta opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS binding
- ChEMBL_603838 (CHEMBL1045633) Agonist activity at human delta opioid receptor expressed in HN9.10 cells assessed as stimulation of [35S]GTPgammaS binding
- ChEMBL_627496 (CHEMBL1111782) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_639784 (CHEMBL1175729) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_639793 (CHEMBL1175738) Antagonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of DPDPE-induced muscle contraction
- ChEMBL_647576 (CHEMBL1217623) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_662964 (CHEMBL1250823) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_699953 (CHEMBL1646360) Antagonist activity at human delta opioid receptor expressed in CHO cells assessed as [35S]GTPgammaS binding by SPA
- ChEMBL_702694 (CHEMBL1657768) Agonist activity at human delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding
- ChEMBL_702698 (CHEMBL1657772) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_736202 (CHEMBL1693238) Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation counting
- ChEMBL_742680 (CHEMBL1769558) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_773196 (CHEMBL1839146) Agonist activity at delta opioid receptor in ICR mouse vas deferens assessed as inhibition of MVD contraction height
- ChEMBL_793549 (CHEMBL1932300) Agonist activity at human recombinant delta opioid receptor expressed in human HEK293 cells by [35S]GTPgammaS binding assay
- ChEMBL_863801 (CHEMBL2175967) Displacement of [3H]DPDPE from delta opioid receptor in calf frontal cortex after 1 hr by gamma counter
- ChEMBL_878872 (CHEMBL2184585) Agonist activity at delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]-GTP-gammaS binding
- ChEMBL_960469 (CHEMBL2389316) Agonist activity at human delta opioid receptor expressed in CHO cells by [35S]GTP-gamma-S binding assay
- ChEMBL_979611 (CHEMBL2424422) Agonist activity at delta opioid receptor in mouse vas deferens assessed as induction of electrically-stimulated muscle contraction
- ChEMBL_979616 (CHEMBL2421108) Antagonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_981013 (CHEMBL2427923) Displacement of [3H]Ile5,6deltorphin-2 from delta opioid receptor in Wistar rat brain membranes by liquid scintillation counting
- ChEMBL_985456 (CHEMBL2432598) Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEBML_153862 In vitro activation of human peroxisome proliferator activated receptor delta (PPAR delta)
- ChEBML_154038 Activity against murine PPAR delta receptor
- ChEBML_145618 Tested for the opioid receptor delta 1 binding affinity using membrane preparations from recombinant HEK293 cells with [3H]naltrindole radioligand
- ChEBML_146485 Compound was evaluated in 3 determinations for the agonistic activity in the Opioid receptor delta 1 of mouse vas deferens
- ChEBML_147160 Binding affinity against Opioid receptor delta 1 of guinea pig brain membranes using 1 nM of [3H]DADLE as radioligand
- ChEBML_1644405 Displacement of [3H]DPDPE from human delta opioid receptor expressed in CHO cell membranes by micro-beta scintillation counting method
- ChEBML_1690602 Displacement of [3H]DADLE from human delta opioid receptor expressed in HEK cells after 90 mins by scintillation counting method
- ChEBML_53447 Binding affinity towards human opioid Delta receptor transfected into Chinese hamster ovary (CHO) cells using [3H]Cl-DPDPE as radioligand.
- ChEBML_53590 Affinity to delta opioid receptor determined in the presence of [3H]- [D-Pen2,5]enkephalin using membranes prepared from rat cerebrum
- ChEMBL_145184 (CHEMBL754284) Binding affinity for Opioid receptor delta 1 by the inhibition of binding of [3H]DADAL in rat brain membranes.
- ChEMBL_145308 (CHEMBL751914) EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor delta 1 (Cl-DPDPE) transfected onto CHO cells
- ChEMBL_145333 (CHEMBL750421) Binding affinity for Opioid receptor delta 1 by the inhibition of binding of [3H]-p-DPDPE human cloned receptors.
- ChEMBL_145483 (CHEMBL751977) Binding affinity towards opioid receptor delta 1 expressed in CHO cells was determined by using [3H]DPDPE as radioligand
- ChEMBL_145769 (CHEMBL752787) Binding affinity was measured in cloned Opioid receptor delta 1 expressed in CHO cells using [3H]- DPDPE as radioligand.
- ChEMBL_146327 (CHEMBL757535) Binding affinity towards opioid receptor delta 1 expressed in CHO cells was determined by using [3H]DPDPE as radioligand
- ChEMBL_146645 (CHEMBL754929) Ability to displace [3H][D-Ser2,Leu5]enkephalin-Thr ([3H]DSLET) from Opioid receptor delta 1 in rat brain
- ChEMBL_146651 (CHEMBL754935) Binding affinity towards delta opioid receptor was determined in rat brain using [H]-[p-Cl-Phe4]-DPDPE as radioligand
- ChEMBL_146653 (CHEMBL754937) Binding potency of compound in competition with [3H]DPDPE for Opioid receptor delta 1 tested in rat brain membrane
- ChEMBL_146756 (CHEMBL753484) Binding affinity for Opioid receptor delta 1 by the inhibition of binding of [3H]DADAL in rat brain membranes.
- ChEMBL_146765 (CHEMBL755209) In vitro inhibition of [3H]- [p-Cl-Phe4]DPDPE binding to Opioid receptor delta 1 using rat brain membranes.
- ChEMBL_147040 (CHEMBL753343) Binding affinity towards Opioid receptor delta 1 was determined in rat brain homogenate using [3H]deltorphin II as radioligand
- ChEMBL_147184 (CHEMBL754483) Opioid receptor delta 1 binding affinity was determined by inhibition of binding of [3H]DADLE to rat brain membrane
- ChEMBL_147280 (CHEMBL755202) Inhibition of [35S]GTP-gamma-S, binding from Opioid receptor delta 1 in Guinea pig Caudate stimulated by SNC80
- ChEMBL_147346 (CHEMBL756190) The compound was tested for binding affinity against Opioid receptor delta 1 by using [3H]- DPDPE as a radioligand
- ChEMBL_1837355 (CHEMBL4337488) Displacement of [3H]DADLE from delta opioid receptor in rat brain after 60 mins by liquid scintillation counting method
- ChEMBL_1906967 (CHEMBL4409325) Inhibition of delta opioid receptor (unknown origin) expressed in human UO5S cells assessed as increase in beta arrestin recruitment
- ChEMBL_1926741 (CHEMBL4429813) Displacement of [125I]-IBNtxA from mouse delta opioid receptor-1 expressed in CHO cell membranes incubated for 90 mins
- ChEMBL_1994961 (CHEMBL4628856) Displacement of [3H]-DPDPE from Wistar rat delta opioid receptor incubated for 3 hrs by liquid scintillation counting method
- ChEMBL_328881 (CHEMBL860461) Agonist potency assessed by [35S]GTP-gammaS binding assay in C6 Glioma cells expressing cloned human delta opioid receptor
- ChEMBL_458382 (CHEMBL942701) Agonist activity at human delta opioid receptor expressed in CHO cell membrane by [35S]GTP-gamma-S binding assay
- ChEMBL_539202 (CHEMBL1024706) Agonist activity at delta opioid receptor in ICR mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_564843 (CHEMBL955070) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation counting
- ChEMBL_717378 (CHEMBL1670100) Displacement of [3H]naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation counting
- ChEMBL_746789 (CHEMBL1777019) Displacement of [3H]naltrindole from human delta-opioid receptor expressed in CHO cells after 3 hrs by scintillation counting
- ChEMBL_793354 (CHEMBL1931908) Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Wistar rat brain membrane by liquid scintillation counting
- ChEMBL_827539 (CHEMBL2051480) Displacement of [3H]DPDPE from delta opioid receptor in rat brain homogenate after 1 hr by liquid scintillation counting
- ChEMBL_839813 (CHEMBL2089824) Displacement of [3H]diprenorphine from human cloned delta type opioid receptor expressed in CHO cell membranes by scintillation counter
- ChEMBL_856456 (CHEMBL2161188) Displacement of [3H]DPDPE from delta-opioid receptor expressed in CHOK1 cells after overnight incubation by scintillation proximity assay
- ChEMBL_859250 (CHEMBL2166335) Agonist activity at delta opioid receptor in Kunming mouse vas deferens assessed as inhibition of electrically-stimulated muscle contraction
- ChEMBL_887195 (CHEMBL2215303) Displacement of [3H]Naltrindole from human delta opioid receptor expressed in CHO cells after 3 hrs by scintillation counting
- ChEMBL_957363 (CHEMBL2378028) Agonist activity at human delta opioid receptor transfected in CHOK1 cells after 60 mins by [35S]GTPgammaS binding assay