Affinity DataKd: 390nMAssay Description:Binding affinity to MDMXMore data for this Ligand-Target Pair
Affinity DataKd: <100nMAssay Description:Tested for antagonist activity at NK-2 tachykinin receptors in hamster tracheaMore data for this Ligand-Target Pair
Affinity DataKd: 84nMAssay Description:Binding affinity towards muscarinic acetylcholine receptor by inhibiting specific binding of [3H]-quinuclidinyl benzilate (0.8 nM) in vitro to membra...More data for this Ligand-Target Pair
Affinity DataKd: 61nMAssay Description:Cross Resistance (antiviral activity) of the compound with Y188C (Nonnucleoside reverse transcriptase inhibitor) resistant HIV isolate from cytopathi...More data for this Ligand-Target Pair
Affinity DataKd: 614nMAssay Description:HIV Protease inhibitory activityMore data for this Ligand-Target Pair
Affinity DataKd: 8.5nMAssay Description:Agonist activity at GPR40 (unknown origin) expressed in mouse A9 cells assessed as inositol phosphate accumulation using [myo-3H]inositol after 1 hr ...More data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Agonist activity at human beta-2 adrenergic receptor expressed in human H292 cells assessed as accumulation of intracellular cAMP after 1 hr by Alpha...More data for this Ligand-Target Pair
Affinity DataKd: 2.30nMAssay Description:Binding affinity to full length human MDM4 by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 221nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Affinity DataKd: 641nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Affinity DataKd: 440nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Affinity DataKd: 279nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Affinity DataKd: 370nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Affinity DataKd: 593nMAssay Description:Binding affinity to MDMX (unknown origin) by using (FITC)-labeled p53 peptide based fluorescence polarization competitive assayMore data for this Ligand-Target Pair
Affinity DataKd: 67nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 187nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 781nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 251nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 372nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 265nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 242nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 115nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 348nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.68E+3nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 570nMAssay Description:Binding affinity to MDMX (unknown origin) by using FITC-labeled compound by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Binding affinity to N-terminal TEV/GST-fused human MDM4 (22 to 110 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation consta...More data for this Ligand-Target Pair
Affinity DataKd: 210nMAssay Description:Tested for its antagonist activity against kappa receptor using U-69,593 as radioligand in isolated guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 229nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Affinity DataKd: 13nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataKd: 43nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
Affinity DataKd: 27nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]; inactive up to a co...More data for this Ligand-Target Pair
Affinity DataKd: 21nMAssay Description:Component deacylation rate constant for interaction with human leukocyte elastaseMore data for this Ligand-Target Pair