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Found 3 of ec50 for monomerid = 29880
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Amgen

LigandPNGBDBM29880(alkynyl ether, 22)
Affinity DataKi:  22nM EC50:  1.40E+3nMAssay Description:The human PPARdelta ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Amgen

LigandPNGBDBM29880(alkynyl ether, 22)
Affinity DataKi:  84nM EC50:  2.20E+3nMAssay Description:The human PPARgamma ligand binding was directly measured using a filtration assay in a UniFilter 350 96-well assay plate (Polyfiltronics). The reacti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Amgen

LigandPNGBDBM29880(alkynyl ether, 22)
Affinity DataKi:  1.90E+3nM ΔG°:  -32.3kJ/mole EC50: >1.00E+5nMpH: 7.1 T: 2°CAssay Description:The human PPARalpha ligand binding was directly measured using a scintillation proximity assay. Plates were read on a Packard TopCount. IC50 values f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed