Compile Data Set for Download or QSAR
maximum 50k data
Found 12 of ec50 for monomerid = 50199176
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human recombinant P2Y2 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human P2Y2 receptor expressed in 1321N1 cells assessed as IP accumulation by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human P2Y6 receptor expressed in 1321N1 cells assessed as IP accumulation by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human recombinant P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production after 30 mins by sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human P2Y6 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 4(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50199176(2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-di...)
Affinity DataEC50:  1.77E+3nMAssay Description:Agonist activity at human P2Y4 receptor expressed in 1321N1 cells assessed as IP accumulation by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed