Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ec50 for monomerid = 50238713
TargetNeuromedin-U receptor 2(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50238713(CHEMBL4070175)
Affinity DataEC50:  0.830nMAssay Description:Agonist activity at human NMUR2 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 2(Mus musculus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50238713(CHEMBL4070175)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at mouse NMUR2 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50238713(CHEMBL4070175)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-U receptor 1(Mus musculus)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50238713(CHEMBL4070175)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at mouse NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed