Affinity DataIC50: 26nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Antagonist activity at P2Y12 receptor in Sprague-Dawley rat platelet rich plasma assessed as inhibition of ADP-induced aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Antagonist activity at P2Y12 receptor in Sprague-Dawley rat platelet rich plasma assessed as inhibition of ADP-induced aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of human coagulation factor 10a using S-2765 as substrate measured up to 20 mins by chromogenic assayMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Antagonist activity at P2Y12 receptor in Sprague-Dawley rat platelet rich plasma assessed as inhibition of ADP-induced aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Antagonist activity at P2Y12 receptor in Sprague-Dawley rat platelet rich plasma assessed as inhibition of ADP-induced aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Antagonist activity at P2Y12 receptor in Sprague-Dawley rat platelet rich plasma assessed as inhibition of ADP-induced aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Antagonist activity at P2Y12 receptor in Sprague-Dawley rat platelet rich plasma assessed as inhibition of ADP-induced aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Antagonist activity at P2Y12 receptor in Sprague-Dawley rat platelet rich plasma assessed as inhibition of ADP-induced aggregationMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of factor-10a (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 86nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 87nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 94nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:Displacement of [33P]2MeS-ADP from P2Y12 receptor (unknown origin) transfected in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Antagonist activity at P2Y12 receptor in Sprague-Dawley rat platelet rich plasma assessed as inhibition of ADP-induced aggregationMore data for this Ligand-Target Pair