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Report error Found 7 of ic50 for monomerid = 119290
LigandPNGBDBM119290(US8673906, 4.09 | US9718800, 4.09)
Affinity DataIC50:  3nMAssay Description:The inhibition of PI3Kβ, PI3Kα, PI3Kγ and PI3Kδ was evaluated in a Kinase Glo based enzyme activity assay using human recombinant...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM119290(US8673906, 4.09 | US9718800, 4.09)
Affinity DataIC50:  3nMT: 25°CAssay Description:Compounds in 100% DMSO were added to assay plates by acoustic dispensing. PI3Kβ was added in a Tris buffer (50 mM Tris pH7.4, 0.05% CHAPS, 2.1 m...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM119290(US8673906, 4.09 | US9718800, 4.09)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant PI3Kbeta using PIP2 by Kinase-Glo Plus assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM119290(US8673906, 4.09 | US9718800, 4.09)
Affinity DataIC50:  17nMAssay Description:Inhibition of PI3Kbeta in PTEN-null human MDA-MB-468 cells assessed as inhibition of Akt phosphorylation after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM119290(US8673906, 4.09 | US9718800, 4.09)
Affinity DataIC50:  90nMAssay Description:Inhibition of human recombinant PI3Kdelta using PIP2 by Kinase-Glo Plus assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM119290(US8673906, 4.09 | US9718800, 4.09)
Affinity DataIC50:  230nMAssay Description:Inhibition of human recombinant PI3Kalpha using PIP2 by Kinase-Glo Plus assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM119290(US8673906, 4.09 | US9718800, 4.09)
Affinity DataIC50:  830nMAssay Description:Inhibition of human recombinant PI3Kgamma using PIP2 by Kinase-Glo Plus assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed