Compile Data Set for Download or QSAR
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Found 5 of ic50 for monomerid = 31543
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM31543(pyrazolo[4,3-h]quinazoline-3-carboxamide, 26)
Affinity DataIC50:  4nMAssay Description:Inhibition of CDK2/Cyclin A2 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D3(Homo sapiens (Human))
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM31543(pyrazolo[4,3-h]quinazoline-3-carboxamide, 26)
Affinity DataIC50:  10nMAssay Description:Inhibition of CDK4/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM31543(pyrazolo[4,3-h]quinazoline-3-carboxamide, 26)
Affinity DataIC50:  24nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Homo sapiens (Human))
Jiangnan University

Curated by ChEMBL
LigandPNGBDBM31543(pyrazolo[4,3-h]quinazoline-3-carboxamide, 26)
Affinity DataIC50:  2.52E+3nMAssay Description:Inhibition of CDK6/Cyclin D3 (unknown origin) using FAM-labeled peptide as substrate after 40 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Nerviano Medical Sciences

LigandPNGBDBM31543(pyrazolo[4,3-h]quinazoline-3-carboxamide, 26)
Affinity DataIC50: >1.00E+4nMT: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates, followed by quantitation of the phosphorylat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed