TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Bristol-Myers
Curated by ChEMBL
Bristol-Myers
Curated by ChEMBL
Affinity DataIC50: 144nMAssay Description:Ability to bind at alpha-2 adrenergic receptor by displacing [3H]clonidineMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Ability to bind at serotonin 5-hydroxytryptamine 1 receptor of rat hippocampus by displacing [3H]5-HTMore data for this Ligand-Target Pair
Affinity DataIC50: 377nMAssay Description:In vitro inhibition of arachidonic acid induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Bristol-Myers
Curated by ChEMBL
Bristol-Myers
Curated by ChEMBL
Affinity DataIC50: 426nMAssay Description:Ability to bind at alpha-1 adrenergic receptor by displacing [3H]WB-4101More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Ability to bind at Dopamine receptor D2 of rat corpus striatum by displacing [3H]spiperoneMore data for this Ligand-Target Pair