Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 50270406
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270406(CHEMBL4084130)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells co-expressing Ric-3/NACHO assessed as inhibition of ACh-induced calcium mobilizat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit beta-2/beta-4(Mus musculus)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270406(CHEMBL4084130)
Affinity DataIC50:  3.00E+4nMAssay Description:Antagonist activity at mouse alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rattus norvegicus (Rat))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50270406(CHEMBL4084130)
Affinity DataIC50: >3.00E+5nMAssay Description:Antagonist activity at rat alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of (S)-nicotine-induced current response measured up to...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed