Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ic50 for monomerid = 50461681
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50461681(Atopaxar | E-5555 | E5555 | ER-172594-00)
Affinity DataIC50:  32nMAssay Description:Antagonist activity at PAR1 in human EAhy926 cells assessed as inhibition of TFLLRN-NH2-induced intracellular calcium mobilization pretreated for 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Marquette University

Curated by ChEMBL
LigandPNGBDBM50461681(Atopaxar | E-5555 | E5555 | ER-172594-00)
Affinity DataIC50:  33nMAssay Description:Antagonist activity at PAR1 in human EAhy926 cells assessed as inhibition of TFLLRN-NH2-induced intracellular calcium mobilization pretreated for 15 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed