TargetCyclin-dependent kinase 7(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: <20nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
Syros Pharmaceuticals
Curated by ChEMBL
Syros Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of CDK9/cyclin T1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assayMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of CDK12/cyclin K (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Syros Pharmaceuticals
Curated by ChEMBL
Syros Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibition of CDK2/cyclin E1 (unknown origin) using 5-FAM-labeled peptide as substrate in presence of ATP by mobility shift assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >200nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Tianjin University of Science and Technology
Curated by ChEMBL
Tianjin University of Science and Technology
Curated by ChEMBL
Affinity DataIC50: >200nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair