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Report error Found 4 of ic50 for monomerid = 9454
TargetAromatase(Human)
Ohio State University

LigandPNGBDBM9454(7-(benzyloxy)-3-phenyl-2-[(pyridin-4-ylmethyl)sulf...)
Affinity DataKi:  220nM ΔG°:  -39.5kJ/mole IC50:  210nMpH: 7.0 T: 37°CAssay Description:Inhibition of human placental aromatase was determined by monitoring the amount of 3H2O released as the enzyme converts [1beta-3H]androst-4-ene-3,17-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Human)
Ohio State University

LigandPNGBDBM9454(7-(benzyloxy)-3-phenyl-2-[(pyridin-4-ylmethyl)sulf...)
Affinity DataIC50:  210nMAssay Description:Inhibition of human placental microsome aromatase using [1beta[3H]]androst-4-ene-3,17-dione as substrate after 15 mins in presence of NADPH by liquid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Human)
Ohio State University

LigandPNGBDBM9454(7-(benzyloxy)-3-phenyl-2-[(pyridin-4-ylmethyl)sulf...)
Affinity DataIC50:  210nMAssay Description:Inhibition of human aromatase-mediated conversion of [1beta3H]androstenedione to estrone by liquid scintillation counting in presence of NADPHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Human)
Ohio State University

LigandPNGBDBM9454(7-(benzyloxy)-3-phenyl-2-[(pyridin-4-ylmethyl)sulf...)
Affinity DataIC50:  2.10E+5nMAssay Description:Inhibition of human placental aromatase assessed as conversion of [1beta-3H]androst-4-ene-3,17-dione to estrone after 15 mins by scintillation counti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed