Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 16132
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Pfizer

LigandPNGBDBM16132(1-guanidino-7-sulfonamidoisoquinoline 6 | 2-(4-chl...)
Affinity DataKi:  140nM ΔG°:  -40.7kJ/molepH: 8.1 T: 2°CAssay Description:Ki values for compounds were calculated by incubation of each enzyme with its substrate and various compound concentrations. Absorbance was read at 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Pfizer

LigandPNGBDBM16132(1-guanidino-7-sulfonamidoisoquinoline 6 | 2-(4-chl...)
Affinity DataKi: >1.00E+5nMAssay Description:Ki values for compounds were calculated by incubation of each enzyme with its substrate and various compound concentrations. Absorbance was read at 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Pfizer

LigandPNGBDBM16132(1-guanidino-7-sulfonamidoisoquinoline 6 | 2-(4-chl...)
Affinity DataKi: >1.00E+5nMAssay Description:Ki values for compounds were calculated by incubation of each enzyme with its substrate and various compound concentrations. Absorbance was read at 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed