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Report error Found 2 of ki for monomerid = 22868
TargetHistamine H1 receptor(Rat)
Schering-Plough

Curated by ChEMBL
LigandPNGBDBM22868(11-(1-methylpiperidin-4-ylidene)-6,11-dihydro-5H-b...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to histamine H1 receptor in rat brain membranes was evaluated using [3H]-pyrilamine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Human)
Vrije Universiteit Amsterdam

LigandPNGBDBM22868(11-(1-methylpiperidin-4-ylidene)-6,11-dihydro-5H-b...)
Affinity DataKi: >1.00E+4nM ΔG°: >-29.7kJ/molepH: 7.4 T: 37°CAssay Description:Ligand displacement assays were performed on The SK-N-MC/hH4R cell homogenates. Retained radioactivity was determined by liquid scintillation countin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed