TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha4-beta2 using +/-[3H]epibatidine as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Displacement of [3H]epibatidine from nAChR alpha4beta2 receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]nicotine from nAChR alpha4beta2 receptorMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit beta-4(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity to Nicotinic acetylcholine receptor alpha3-beta4 using +/-[3H]epibatidine as radioligand in pig adrenal glandMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity to subtype Nicotinic acetylcholine receptor alpha7 using [3H]-MLA as radioligand in rat brainMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Institut F£R Pharmazeutische Chemie Der Philipps-Universit£T Marburg
Curated by ChEMBL
Affinity DataKi: 2.76E+3nMAssay Description:Binding affinity at rat brain Nicotinic acetylcholine receptor alpha7More data for this Ligand-Target Pair