Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ki for monomerid = 50542790
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50542790(CHEMBL4647584)
Affinity DataKi:  0.130nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 120 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50542790(CHEMBL4647584)
Affinity DataKi:  0.490nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 30 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50542790(CHEMBL4647584)
Affinity DataKi:  0.620nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 90 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50542790(CHEMBL4647584)
Affinity DataKi:  0.730nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 60 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetN-terminal Xaa-Pro-Lys N-methyltransferase 1(Homo sapiens)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50542790(CHEMBL4647584)
Affinity DataKi:  15nMAssay Description:Time dependent inhibition of NTMT1 (unknown origin) pre-incubated for 10 mins before GPKRIA peptide substrate addition by SAHH coupled fluorescence a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed