TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Helmholtz Centre For Infection Research
Curated by ChEMBL
Helmholtz Centre For Infection Research
Curated by ChEMBL
Affinity DataKd: 7nMAssay Description:Binding affinity to human PPARgamma (unknown origin) by competitive TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Helmholtz Centre For Infection Research
Curated by ChEMBL
Helmholtz Centre For Infection Research
Curated by ChEMBL
Affinity DataKd: 14.8nM EC50: 3.80nMpH: 7.5 T: 2°CAssay Description:Kd values were obtained by incubating His-PPARgamma-LBD with biotinylated peptide, europium-labeled anti-histidine antibody, and allophycocyanin-labe...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Helmholtz Centre For Infection Research
Curated by ChEMBL
Helmholtz Centre For Infection Research
Curated by ChEMBL
Affinity DataKd: 120nMAssay Description:Binding affinity to PPARgamma ligand binding domain by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Helmholtz Centre For Infection Research
Curated by ChEMBL
Helmholtz Centre For Infection Research
Curated by ChEMBL
Affinity DataKd: 4.98E+3nMAssay Description:Binding affinity to human PPARgammaMore data for this Ligand-Target Pair