Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of kd for monomerid = 50585045
LigandPNGBDBM50585045(CHEMBL5093741)
Affinity DataKd:  0.912nMAssay Description:Binding affinity to human DYRK1A assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
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TargetDual specificity protein kinase CLK1(Homo sapiens (Human))TBA
LigandPNGBDBM50585045(CHEMBL5093741)
Affinity DataKd:  35nMAssay Description:Binding affinity to human CLK1 assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))TBA
LigandPNGBDBM50585045(CHEMBL5093741)
Affinity DataKd:  7.29E+3nMAssay Description:Binding affinity to human GSK-3beta assessed as equilibrium dissociation constant measured upto 240 min by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed