Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of kd for monomerid = 50601440
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50601440(CHEMBL5176837)
Affinity DataKd:  0.0100nMAssay Description:Binding affinity to FLT3-ITD-D835V mutant (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50601440(CHEMBL5176837)
Affinity DataKd:  0.290nMAssay Description:Binding affinity to FLT3-TKD-D835V mutant (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50601440(CHEMBL5176837)
Affinity DataKd:  0.290nMAssay Description:Binding affinity to FLT3-TKD-D835H mutant (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50601440(CHEMBL5176837)
Affinity DataKd:  0.290nMAssay Description:Binding affinity to FLT3-TKD-D835Y mutant (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50601440(CHEMBL5176837)
Affinity DataKd:  0.300nMAssay Description:Binding affinity to FLT3-R834Q mutant (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50601440(CHEMBL5176837)
Affinity DataKd:  0.330nMAssay Description:Binding affinity to FLT3-N841I mutant (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50601440(CHEMBL5176837)
Affinity DataKd:  0.360nMAssay Description:Binding affinity to FLT3-ITD (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50601440(CHEMBL5176837)
Affinity DataKd:  5.40nMAssay Description:Binding affinity to FLT3-K663Q mutant (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails PubMed