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Found 142 Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 1'
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157676(CHEMBL426565 | N-(2,6-diphenylpyrimidin-4-yl)aceta...)
Affinity DataKi:  31.2nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157663(CHEMBL222718 | N-(4,6-diphenylpyrimidin-2-yl)propi...)
Affinity DataKi:  31.3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335726(CHEMBL1650371 | N-2,6-bis2-methoxyphenyl)pyrimidin...)
Affinity DataKi:  31.6nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335746(CHEMBL1650398 | N-(2,6-bis(4-methoxyphenyl)pyrimid...)
Affinity DataKi:  32.1nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335739(CHEMBL1650388 | N-2,6-dithiophen-2-yl)pyrimidin-4-...)
Affinity DataKi:  32.9nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335740(CHEMBL1650389 | N-2,6-dithiophen-2-yl)pyrimidin-4-...)
Affinity DataKi:  33.3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335721(CHEMBL1650366 | N-2,6-bis4-fluorophenyl)pyrimidin-...)
Affinity DataKi:  34.8nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335708(CHEMBL1650350 | N-2,6-di-p-tolylpyrimidin-4-yl)pro...)
Affinity DataKi:  36.9nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335699(CHEMBL1650394 | N-2,6-dithiophen-3-yl)pyrimidin-4-...)
Affinity DataKi:  39.4nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335741(CHEMBL1650393 | N-2,6-dithiophen-3-yl)pyrimidin-4-...)
Affinity DataKi:  39.8nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335694(CHEMBL1650384 | N-2,6-difuran-2-yl)pyrimidin-4-yl)...)
Affinity DataKi:  40.7nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335730(CHEMBL1650375 | N-2,6-bis2-fluorophenyl)pyrimidin-...)
Affinity DataKi:  41.3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157663(CHEMBL222718 | N-(4,6-diphenylpyrimidin-2-yl)propi...)
Affinity DataKi:  42.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335715(CHEMBL1650359 | N-2,6-bis4-methylthio)phenyl)pyrim...)
Affinity DataKi:  43.6nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335717(CHEMBL1650362 | N-2,6-bis4-acetylphenyl)pyrimidin-...)
Affinity DataKi:  43.9nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  45.5nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335737(CHEMBL1650383 | N-2,6-distyrylpyrimidin-4-yl)propi...)
Affinity DataKi:  46.9nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335700(CHEMBL1650142 | N-(4,6-dip-tolylpyrimidin-2-yl)ace...)
Affinity DataKi:  47.3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335690(CHEMBL1650164 | N-(4,6-bis(2-methoxyphenyl)pyrimid...)
Affinity DataKi:  48.2nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335698(CHEMBL1650391 | N-2,6-difuran-3-yl)pyrimidin-4-yl)...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335748(CHEMBL1650400 | N-(2,6-bis(2,4-dimethoxyphenyl)pyr...)
Affinity DataKi:  52.4nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335749(CHEMBL1650401 | N-(2,6-bis(2,4-dimethoxyphenyl)pyr...)
Affinity DataKi:  56.3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335745(CHEMBL1650397 | N-(2,6-bis(4-methoxyphenyl)pyrimid...)
Affinity DataKi:  58.1nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335735(CHEMBL1650381 | N-2,6-dibenzo[d][1,3]dioxol-6-yl)p...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335709(CHEMBL1650351 | N-2,6-di-p-tolylpyrimidin-4-yl)but...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335722(CHEMBL1650367 | N-2,6-bis4-chlorophenyl)pyrimidin-...)
Affinity DataKi:  63.3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335699(CHEMBL1650394 | N-2,6-dithiophen-3-yl)pyrimidin-4-...)
Affinity DataKi:  63.5nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335699(CHEMBL1650394 | N-2,6-dithiophen-3-yl)pyrimidin-4-...)
Affinity DataKi:  64.2nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335752(CHEMBL1650395 | N-2,6-dithiophen-3-yl)pyrimidin-4-...)
Affinity DataKi:  65.1nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335751(CHEMBL1650392 | N-2,6-difuran-3-yl)pyrimidin-4-yl)...)
Affinity DataKi:  65.1nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335714(CHEMBL1650358 | N-2,6-bis4-methylthio)phenyl)pyrim...)
Affinity DataKi:  71.3nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335725(CHEMBL1650370 | N-2,6-bis2-methoxyphenyl)pyrimidin...)
Affinity DataKi:  73.8nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335697(CHEMBL1650390 | N-2,6-difuran-3-yl)pyrimidin-4-yl)...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  76.6nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335721(CHEMBL1650366 | N-2,6-bis4-fluorophenyl)pyrimidin-...)
Affinity DataKi:  82.3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335698(CHEMBL1650391 | N-2,6-difuran-3-yl)pyrimidin-4-yl)...)
Affinity DataKi:  82.8nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335720(CHEMBL1650365 | N-2,6-bis4-fluorophenyl)pyrimidin-...)
Affinity DataKi:  83.9nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157672(CHEMBL222474 | N-(2,6-diphenylpyrimidin-4-yl)propi...)
Affinity DataKi:  84.5nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335743(CHEMBL1650348 | N-(4,6-di(thiophen-3-yl)pyrimidin-...)
Affinity DataKi:  85.7nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335702(CHEMBL1650172 | N-(4,6-di(benzo[d][1,3]dioxol-5-yl...)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335726(CHEMBL1650371 | N-2,6-bis2-methoxyphenyl)pyrimidin...)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335724(CHEMBL1650369 | N-2,6-bis4-chlorophenyl)pyrimidin-...)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50157659(CHEMBL222384 | N-(2,6-diphenylpyrimidin-4-yl)butyr...)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335730(CHEMBL1650375 | N-2,6-bis2-fluorophenyl)pyrimidin-...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335729(CHEMBL1650374 | N-2,6-bis2-fluorophenyl)pyrimidin-...)
Affinity DataKi:  113nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335739(CHEMBL1650388 | N-2,6-dithiophen-2-yl)pyrimidin-4-...)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]ZM2413853 from human adenosine A2A receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335710(CHEMBL1650352 | N-2,6-bis4-trifluoromethyl)phenyl)...)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335692(CHEMBL1650173 | N-(4,6-di(benzo[d][1,3]dioxol-5-yl...)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335688(CHEMBL1650144 | N-(4,6-dip-tolylpyrimidin-2-yl)but...)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in human HeLa cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50335698(CHEMBL1650391 | N-2,6-difuran-3-yl)pyrimidin-4-yl)...)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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