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Found 184 Enz. Inhib. hit(s) with all data for entry = 50004866
LigandPNGBDBM21792(2-[(1S)-5-{3-[4-(4-tert-butyl-1,3-thiazol-2-yl)-2-...)
Affinity DataEC50:  9.09E+7nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21824(2-[(1S)-5-{3-[4-(4-ethoxy-5-methyl-1,3-thiazol-2-y...)
Affinity DataEC50:  1.67E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21812(2-[4-(3-{[(1S)-1-(carboxymethyl)-2,3-dihydro-1H-in...)
Affinity DataEC50:  4.27E+6nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21777(2-[(1S)-5-(3-{2-methyl-4-[3-(trifluoromethyl)-1,2,...)
Affinity DataEC50:  1.92E+6nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM21776(2-[(1S)-5-{3-[2-chloro-4-(4H-1,2,4-triazol-4-yl)ph...)
Affinity DataEC50:  4.48E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM21789(2-[(1S)-5-{3-[4-(4-ethyl-1,3-thiazol-2-yl)phenoxy]...)
Affinity DataEC50:  7.81E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21814(2-[4-(3-{[(1S)-1-(carboxymethyl)-2,3-dihydro-1H-in...)
Affinity DataEC50:  1.15E+6nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21792(2-[(1S)-5-{3-[4-(4-tert-butyl-1,3-thiazol-2-yl)-2-...)
Affinity DataEC50:  5.62E+7nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21763(2-[(1S)-5-{3-[4-(pyrimidin-5-yl)phenoxy]propoxy}-2...)
Affinity DataEC50:  1.05E+6nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21774(2-[(1S)-5-{3-[4-(1H-1,2,4-triazol-1-yl)phenoxy]pro...)
Affinity DataEC50:  1.82E+6nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM21761(2-[(1S)-5-[3-(3-methylphenoxy)propoxy]-2,3-dihydro...)
Affinity DataEC50:  1.26E+5nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21819(2-[(1S)-5-{3-[4-(4-ethoxy-1,3-thiazol-2-yl)-2-prop...)
Affinity DataEC50:  5.00E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21804(2-[(1S)-5-[3-(2-methoxy-4-{5H,6H,7H-pyrano[2,3-d][...)
Affinity DataEC50:  7.69E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21797(2-[(1S)-5-[3-(4-{4H,5H,6H-cyclopenta[d][1,3]thiazo...)
Affinity DataEC50:  7.69E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21788(2-[(1S)-5-{3-[2-methoxy-4-(4-methyl-1,3-thiazol-2-...)
Affinity DataEC50:  3.70E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21767(2-[(1S)-5-{3-[2-propyl-4-(trifluoromethyl)phenoxy]...)
Affinity DataEC50:  8.77E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21808(2-[(1S)-5-{3-[4-(5-acetyl-4-methyl-1,3-thiazol-2-y...)
Affinity DataEC50:  1.79E+6nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21795(2-[(1S)-5-{3-[4-(4,5-dimethyl-1,3-thiazol-2-yl)phe...)
Affinity DataEC50:  8.00E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21780(2-[(1S)-5-{3-[4-(1H-indol-6-yl)phenoxy]propoxy}-2,...)
Affinity DataEC50:  1.52E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21771(2-[(1S)-5-[3-(4-ethyl-2-methoxyphenoxy)propoxy]-2,...)
Affinity DataEC50:  3.70E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21761(2-[(1S)-5-[3-(3-methylphenoxy)propoxy]-2,3-dihydro...)
Affinity DataEC50:  1.79E+7nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21823(2-[(1S)-5-{3-[4-(4-ethoxy-5-methyl-1,3-thiazol-2-y...)
Affinity DataEC50:  1.64E+7nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21781(2-[(1S)-5-{3-[4-(pyridin-3-yl)phenoxy]propoxy}-2,3...)
Affinity DataEC50:  1.82E+6nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21818(2-[(1S)-5-{3-[4-(4-ethoxy-1,3-thiazol-2-yl)phenoxy...)
Affinity DataEC50:  1.00E+7nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21763(2-[(1S)-5-{3-[4-(pyrimidin-5-yl)phenoxy]propoxy}-2...)
Affinity DataEC50:  1.37E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21818(2-[(1S)-5-{3-[4-(4-ethoxy-1,3-thiazol-2-yl)phenoxy...)
Affinity DataEC50:  8.33E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21756(2-[(1S)-5-{3-[4-(trifluoromethoxy)phenoxy]propoxy}...)
Affinity DataEC50:  1.00E+6nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21775(2-[(1S)-5-{3-[2-acetamido-4-(1H-1,2,3-triazol-1-yl...)
Affinity DataEC50:  2.72E+6nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
LigandPNGBDBM21781(2-[(1S)-5-{3-[4-(pyridin-3-yl)phenoxy]propoxy}-2,3...)
Affinity DataEC50:  4.35E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21813(2-[4-(3-{[(1S)-1-(carboxymethyl)-2,3-dihydro-1H-in...)
Affinity DataEC50:  1.00E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21779(2-[(1S)-5-{3-[4-(furan-3-yl)phenoxy]propoxy}-2,3-d...)
Affinity DataEC50:  3.06E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21807(2-[(1S)-5-{3-[4-(5-acetyl-4-methyl-1,3-thiazol-2-y...)
Affinity DataEC50:  5.89E+7nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21796(2-[(1S)-5-{3-[4-(4,5-dimethyl-1,3-thiazol-2-yl)-2-...)
Affinity DataEC50:  2.50E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21780(2-[(1S)-5-{3-[4-(1H-indol-6-yl)phenoxy]propoxy}-2,...)
Affinity DataEC50:  6.67E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21790(2-[(1S)-5-{3-[4-(4-ethyl-1,3-thiazol-2-yl)-2-propy...)
Affinity DataEC50:  2.24E+7nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21754(2-[(1S)-5-[3-(4-ethylphenoxy)propoxy]-2,3-dihydro-...)
Affinity DataEC50:  1.62E+5nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21807(2-[(1S)-5-{3-[4-(5-acetyl-4-methyl-1,3-thiazol-2-y...)
Affinity DataEC50:  5.56E+7nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21755(2-[(1S)-5-{3-[4-(trifluoromethyl)phenoxy]propoxy}-...)
Affinity DataEC50:  1.82E+5nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21822(2-[(1S)-5-(3-{2-methoxy-4-[4-(propan-2-yloxy)-1,3-...)
Affinity DataEC50:  3.33E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21817(2-[(1S)-5-{3-[2-methoxy-4-(4-methoxy-1,3-thiazol-2...)
Affinity DataEC50:  3.33E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21805(2-[(1S)-5-{3-[4-(1,3-benzothiazol-2-yl)-2-methoxyp...)
Affinity DataEC50:  1.92E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21800(2-[(1S)-5-{3-[4-(4,5,6,7-tetrahydro-1,3-benzothiaz...)
Affinity DataEC50:  4.55E+8nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARdelta ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21805(2-[(1S)-5-{3-[4-(1,3-benzothiazol-2-yl)-2-methoxyp...)
Affinity DataEC50:  1.90E+6nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21800(2-[(1S)-5-{3-[4-(4,5,6,7-tetrahydro-1,3-benzothiaz...)
Affinity DataEC50:  2.56E+6nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21788(2-[(1S)-5-{3-[2-methoxy-4-(4-methyl-1,3-thiazol-2-...)
Affinity DataEC50:  3.73E+6nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21781(2-[(1S)-5-{3-[4-(pyridin-3-yl)phenoxy]propoxy}-2,3...)
Affinity DataEC50:  5.92E+5nMAssay Description:Agonist activity at GST-tagged Homo sapiens (human) PPARalpha ligand binding domain after 2 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21825(2-[(1S)-5-{3-[4-(4-ethoxy-5-ethyl-1,3-thiazol-2-yl...)
Affinity DataEC50:  5.62E+6nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21819(2-[(1S)-5-{3-[4-(4-ethoxy-1,3-thiazol-2-yl)-2-prop...)
Affinity DataEC50:  2.45E+7nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21813(2-[4-(3-{[(1S)-1-(carboxymethyl)-2,3-dihydro-1H-in...)
Affinity DataEC50:  1.00E+6nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM21808(2-[(1S)-5-{3-[4-(5-acetyl-4-methyl-1,3-thiazol-2-y...)
Affinity DataEC50:  2.04E+7nMAssay Description:Agonist activity at Homo sapiens (human) PPARgamma expressed in mouse 3T3-L1 cells incubated for 2 days followed by compound wash out measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
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