Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50005559
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 0.0500nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of temperature-induced calcium flux after 30 mins by Fluo...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of capsaicin-induced calcium flux after 30 mins by Fluo-4...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of temperature-induced calcium flux after 30 mins by Fluo...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 0.180nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of capsaicin-induced calcium flux after 30 mins by Fluo-4...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 0.290nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of temperature-induced calcium flux after 30 mins by Fluo...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 0.330nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of capsaicin-induced calcium flux after 30 mins by Fluo-4...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 0.340nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of capsaicin-induced calcium flux after 30 mins by Fluo-4...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 0.770nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of capsaicin-induced calcium flux after 30 mins by Fluo-4...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of temperature-induced calcium flux after 30 mins by Fluo...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of temperature-induced calcium flux after 30 mins by Fluo...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of capsaicin-induced calcium flux after 30 mins by Fluo-4...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of temperature-induced calcium flux after 30 mins by Fluo...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of capsaicin-induced calcium flux after 30 mins by Fluo-4...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of capsaicin-induced calcium flux after 30 mins by Fluo-4...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
University of Concepcion
Curated by ChEMBL
University of Concepcion
Curated by ChEMBL
Affinity DataIC50: 6.10nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in HEK293T cells assessed as inhibition of capsaicin-induced calcium flux after 30 mins by Fluo-4...More data for this Ligand-Target Pair