TargetHistone deacetylase 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human His tagged HDAC1 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human His tagged HDAC1 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human His tagged HDAC1 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant human His tagged HDAC1 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 136nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 139nMAssay Description:Inhibition of recombinant human HDAC2 assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 144nMAssay Description:Inhibition of recombinant human HDAC2 assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human His tagged HDAC1 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 205nMAssay Description:Inhibition of recombinant human HDAC2 assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 215nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 234nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 274nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Inhibition of recombinant human HDAC2 assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 381nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 441nMAssay Description:Inhibition of recombinant human HDAC2 assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of recombinant human His tagged HDAC1 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of recombinant human HDAC2 assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins followed by subs...More data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 7.23E+3nMAssay Description:Inhibition of recombinant human His tagged HDAC6 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human His tagged HDAC6 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human HDAC8 assessed as decrease in deacetylation of FLUOR DE LYS substrate preincubated for 10 mins followed by substrate ...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human HDAC8 assessed as decrease in deacetylation of FLUOR DE LYS substrate preincubated for 10 mins followed by substrate ...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human His tagged HDAC6 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human HDAC8 assessed as decrease in deacetylation of FLUOR DE LYS substrate preincubated for 10 mins followed by substrate ...More data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract assessed as decrease in deacetylation of FLUOR DE LYS Green substrate preincubated for 10 mins ...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human HDAC8 assessed as decrease in deacetylation of FLUOR DE LYS substrate preincubated for 10 mins followed by substrate ...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human HDAC8 assessed as decrease in deacetylation of FLUOR DE LYS substrate preincubated for 10 mins followed by substrate ...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human His tagged HDAC6 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human His tagged HDAC6 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetNuclear receptor corepressor 1(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human HDAC3/NCOR1 assessed as decrease in deacetylation of FLUOR DE LYS SIRT1 substrate preincubated for 10 mins followed b...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human His tagged HDAC6 expressed in baculovirus infected insect cells assessed as decrease in deacetylation of FLUOR DE LYS...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Beijing University of Chemical Technology
Curated by ChEMBL
Beijing University of Chemical Technology
Curated by ChEMBL
Affinity DataIC50: >3.20E+4nMAssay Description:Inhibition of recombinant human HDAC8 assessed as decrease in deacetylation of FLUOR DE LYS substrate preincubated for 10 mins followed by substrate ...More data for this Ligand-Target Pair
![](/img/powered_by_small.gif)