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Found 45 Enz. Inhib. hit(s) with all data for entry = 50018099
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403302(CHEMBL5290323)
Affinity DataKi:  6.80nMAssay Description:Tested for its antagonist activity against mu receptor using DAMGO as radioligand in isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403372(CHEMBL5286157)
Affinity DataKi:  7.70nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403372(CHEMBL5286157)
Affinity DataKi:  25nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50014089(CHEMBL1236726)
Affinity DataKi:  109nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403369(CHEMBL5271133)
Affinity DataKi:  620nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403369(CHEMBL5271133)
Affinity DataKi:  620nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50436047(CHEMBL1233798)
Affinity DataKi:  916nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403368(CHEMBL5290720)
Affinity DataKi:  5.50E+3nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50014089(CHEMBL1236726)
Affinity DataKi:  1.10E+4nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50436047(CHEMBL1233798)
Affinity DataKi:  3.60E+4nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403369(CHEMBL5271133)
Affinity DataKi:  5.40E+4nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403368(CHEMBL5290720)
Affinity DataKi:  5.40E+4nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50229787((4S,5R)-Nutlin-3 | (rac)-(4,5-bis(4-chlorophenyl)-...)
Affinity DataKi:  6.90E+4nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50229787((4S,5R)-Nutlin-3 | (rac)-(4,5-bis(4-chlorophenyl)-...)
Affinity DataKi:  7.00E+4nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM6863(US8815926, 101 | US8815926, 295)
Affinity DataIC50:  0.210nMAssay Description:Antagonist activity at NK-2 tachykinin receptors in rabbit pulmonary arteryMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM6863(US8815926, 101 | US8815926, 295)
Affinity DataIC50:  0.210nMAssay Description:Tested for inhibitory activity against (DPDE)delta receptor in mouse vas deferensMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403302(CHEMBL5290323)
Affinity DataIC50:  0.900nMAssay Description:Tested for its antagonist activity against mu receptor using DAMGO as radioligand in isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403528(CHEMBL5280843)
Affinity DataIC50:  17nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]; inactive up to a co...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403525(CHEMBL3220312)
Affinity DataIC50:  17nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50229787((4S,5R)-Nutlin-3 | (rac)-(4,5-bis(4-chlorophenyl)-...)
Affinity DataIC50:  19nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50261656(CHEMBL3347578)
Affinity DataIC50:  20nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403525(CHEMBL3220312)
Affinity DataIC50:  25nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403482(CHEMBL5267044)
Affinity DataIC50:  33nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50261656(CHEMBL3347578)
Affinity DataIC50:  40nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403482(CHEMBL5267044)
Affinity DataIC50:  41nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403303(CHEMBL5273706)
Affinity DataIC50:  44nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403304(CHEMBL5268770)
Affinity DataIC50:  110nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403529(CHEMBL5290391)
Affinity DataIC50:  145nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403303(CHEMBL5273706)
Affinity DataIC50:  550nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM6863(US8815926, 101 | US8815926, 295)
Affinity DataIC50:  3.00E+3nMAssay Description:Tested for its antagonist activity against kappa receptor using U-69,593 as radioligand in isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403530(CHEMBL5267194)
Affinity DataIC50:  3.70E+3nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]; inactive up to a co...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403530(CHEMBL5267194)
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity at NK-2 tachykinin receptors in rabbit pulmonary arteryMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403305(CHEMBL5275075)
Affinity DataKd:  216nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403527(CHEMBL5280949)
Affinity DataKd:  27nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]; inactive up to a co...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403526(CHEMBL5286722)
Affinity DataEC50:  2.60E+4nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403526(CHEMBL5286722)
Affinity DataEC50:  2.30E+3nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403301(CHEMBL4289676)
Affinity DataKd:  210nMAssay Description:Tested for its antagonist activity against kappa receptor using U-69,593 as radioligand in isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403367(CHEMBL5283428)
Affinity DataKd:  43nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403367(CHEMBL5283428)
Affinity DataKd:  25nMAssay Description:Antagonistic activity against M3 muscarinic receptor in guinea pig left ileum derived by plotting log(DR - 1) vs log[antagonist]More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50437206(CHEMBL2402737)
Affinity DataKd: <100nMAssay Description:Tested for antagonist activity at NK-2 tachykinin receptors in hamster tracheaMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403367(CHEMBL5283428)
Affinity DataKd:  149nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403306(CHEMBL5271788)
Affinity DataKd:  13nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein Mdm4(Homo sapiens (Human))TBA
LigandPNGBDBM50403305(CHEMBL5275075)
Affinity DataKd:  229nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403306(CHEMBL5271788)
Affinity DataKd:  12nMAssay Description:Tested for ability to inhibit human erythrocyte carbonic-anhydrase-II- (HCA II) catalyzed carbon dioxide hydrationMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))TBA
LigandPNGBDBM50403301(CHEMBL4289676)
Affinity DataKd:  600nMAssay Description:Tested for its antagonist activity against (DPDE)delta receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails PubMed