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Found 19 Enz. Inhib. hit(s) with all data for entry = 50018283
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50410642(CHEMBL5287722)
Affinity DataIC50:  0.180nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50410643(CHEMBL5289030)
Affinity DataIC50:  0.340nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50410568(CHEMBL5287991)
Affinity DataIC50:  0.510nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)
Affinity DataIC50:  0.600nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenate at pH 9.0More data for this Ligand-Target Pair
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50324574((R)-6-Methoxy-N-(2-((1-methylpiperidin-4-yl)methox...)
Affinity DataIC50: <1nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM412136(US10392402, Compound A | US10738007, Compound A | ...)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
Ligand InfoPurchaseMCE
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TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50410568(CHEMBL5287991)
Affinity DataIC50:  1.20nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM14047(Aminofurazanyl-azabenzimidazole 6n | N-(3-{[2-(4-a...)
Affinity DataIC50:  1.60nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50319005((R)-4-(1-aminoethyl)-N-(1H-pyrrolo[2,3-b]pyridin-4...)
Affinity DataIC50:  3.60nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50319005((R)-4-(1-aminoethyl)-N-(1H-pyrrolo[2,3-b]pyridin-4...)
Affinity DataIC50:  3.60nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM14047(Aminofurazanyl-azabenzimidazole 6n | N-(3-{[2-(4-a...)
Affinity DataIC50:  4nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50410567(CHEMBL5266198)
Affinity DataIC50:  19nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50410567(CHEMBL5266198)
Affinity DataIC50:  19nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50410783(BELUMOSUDIL)
Affinity DataIC50:  105nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50027431(HYDROXYFASUDIL | Hydroxy-Fasudil)
Affinity DataIC50:  720nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50027431(HYDROXYFASUDIL | Hydroxy-Fasudil)
Affinity DataIC50:  720nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50410569(CHEMBL5278924)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50410569(CHEMBL5278924)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
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TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50410783(BELUMOSUDIL)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibitory activity against FAAH in Wistar rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails PubMed