Affinity DataKi: <0.0100nMAssay Description:Binding affinity to Bcl-2 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Binding affinity to recombinant His-tagged human Bcl-xL expressed in Escherichia coli assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Binding affinity to recombinant His-tagged human Bcl-2 expressed in Escherichia coli assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity to recombinant His-tagged human Bcl-2 expressed in Escherichia coli assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity to recombinant His-tagged human Bcl-xL expressed in Escherichia coli assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Binding affinity to Bcl-2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity to Bcl-xL (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 245nMAssay Description:Binding affinity to Bcl-w (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Inhibition of Flu-BakBH3 binding to Bcl-2 (unknown origin) assessed as inhibition constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: >444nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:Binding affinity to Bcl-xL (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of BH3 peptide binding to Mcl-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Inhibition of BH3 peptide binding to Bcl-xL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Inhibition of BH3 peptide binding to Bcl-2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 620nMAssay Description:Inhibition of BH3 peptide binding to Bfl-1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of Bcl-2 (unknown origin) by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.27E+3nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by ELISA analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of Flu-BakBH3 binding to recombinant GST-tagged Bcl-2 (unknown origin) incubated for 30 mins by competitive fluorescence polarization assa...More data for this Ligand-Target Pair
Affinity DataKd: 3.61E+4nMAssay Description:Binding affinity to recombinant Bcl-2 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by MST analys...More data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+3nMAssay Description:Inhibition of Flu-BakBH3 binding to GST-tagged Bcl-2 (unknown origin) preincubated for 10 mins followed by Flu-BakBH3 addition and measured after 30 ...More data for this Ligand-Target Pair