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Found 21 Enz. Inhib. hit(s) with all data for entry = 50018493
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50162774(ABT-199 | US11420968, Example ABT-199 | Venetoclax)
Affinity DataKi: <0.0100nMAssay Description:Binding affinity to Bcl-2 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
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TargetBcl-2-like protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50558853(CHEMBL4465826)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to recombinant His-tagged human Bcl-xL expressed in Escherichia coli assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50608721(CHEMBL5283370)
Affinity DataKi:  9.5nMAssay Description:Binding affinity to recombinant His-tagged human Bcl-2 expressed in Escherichia coli assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50558853(CHEMBL4465826)
Affinity DataKi:  17nMAssay Description:Binding affinity to recombinant His-tagged human Bcl-2 expressed in Escherichia coli assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBcl-2-like protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608722(CHEMBL5278443)
Affinity DataKi:  22nMAssay Description:Binding affinity to recombinant His-tagged human Bcl-xL expressed in Escherichia coli assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50608723(CHEMBL5285186)
Affinity DataKi:  25nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50608723(CHEMBL5285186)
Affinity DataKi:  35nMAssay Description:Binding affinity to Bcl-2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBcl-2-like protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50162774(ABT-199 | US11420968, Example ABT-199 | Venetoclax)
Affinity DataKi:  48nMAssay Description:Binding affinity to Bcl-xL (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
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TargetBcl-2-like protein 2(Homo sapiens (Human))TBA
LigandPNGBDBM50162774(ABT-199 | US11420968, Example ABT-199 | Venetoclax)
Affinity DataKi:  245nMAssay Description:Binding affinity to Bcl-w (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
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TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKi:  320nMAssay Description:Inhibition of Flu-BakBH3 binding to Bcl-2 (unknown origin) assessed as inhibition constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
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LigandPNGBDBM50162774(ABT-199 | US11420968, Example ABT-199 | Venetoclax)
Affinity DataKi: >444nMAssay Description:Binding affinity to Mcl-1 (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
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TargetBcl-2-like protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608723(CHEMBL5285186)
Affinity DataKi:  660nMAssay Description:Binding affinity to Bcl-xL (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50316672((R)-1,1',6,6',7,7'-Hexahydroxy-3,3'-dimethyl-N5-((...)
Affinity DataIC50:  200nMAssay Description:Inhibition of BH3 peptide binding to Mcl-1 (unknown origin)More data for this Ligand-Target Pair
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TargetBcl-2-like protein 1(Homo sapiens (Human))TBA
LigandPNGBDBM50316672((R)-1,1',6,6',7,7'-Hexahydroxy-3,3'-dimethyl-N5-((...)
Affinity DataIC50:  310nMAssay Description:Inhibition of BH3 peptide binding to Bcl-xL (unknown origin)More data for this Ligand-Target Pair
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TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50316672((R)-1,1',6,6',7,7'-Hexahydroxy-3,3'-dimethyl-N5-((...)
Affinity DataIC50:  320nMAssay Description:Inhibition of BH3 peptide binding to Bcl-2 (unknown origin)More data for this Ligand-Target Pair
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TargetBcl-2-related protein A1(Homo sapiens (Human))TBA
LigandPNGBDBM50316672((R)-1,1',6,6',7,7'-Hexahydroxy-3,3'-dimethyl-N5-((...)
Affinity DataIC50:  620nMAssay Description:Inhibition of BH3 peptide binding to Bfl-1 (unknown origin)More data for this Ligand-Target Pair
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TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50505361(CHEMBL4530348)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of Bcl-2 (unknown origin) by ELISA analysisMore data for this Ligand-Target Pair
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TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50234313(CHEMBL4102399)
Affinity DataIC50:  4.27E+3nMAssay Description:Binding affinity to Bcl-2 (unknown origin) by ELISA analysisMore data for this Ligand-Target Pair
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TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50200965(2-Amino-6-bromo-4-(cyano-ethoxycarbonyl-methyl)-4H...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of Flu-BakBH3 binding to recombinant GST-tagged Bcl-2 (unknown origin) incubated for 30 mins by competitive fluorescence polarization assa...More data for this Ligand-Target Pair
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TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50412286(CHEMBL476730)
Affinity DataKd:  3.61E+4nMAssay Description:Binding affinity to recombinant Bcl-2 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constant by MST analys...More data for this Ligand-Target Pair
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TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM31802(Apogossypol | US9115061, Apogossypol)
Affinity DataEC50:  2.80E+3nMAssay Description:Inhibition of Flu-BakBH3 binding to GST-tagged Bcl-2 (unknown origin) preincubated for 10 mins followed by Flu-BakBH3 addition and measured after 30 ...More data for this Ligand-Target Pair
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