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Found 64 Enz. Inhib. hit(s) with all data for entry = 50018626
TargetMacrophage metalloelastase(Homo sapiens (Human))TBA
LigandPNGBDBM50433864(CHEMBL2380403)
Affinity DataKi:  4.80nMAssay Description:Inhibition of MMP12 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))TBA
LigandPNGBDBM50433864(CHEMBL2380403)
Affinity DataKi:  5nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50264810(CHEMBL445971 | N-(4-(4-(thiiran-2-ylmethylsulfonyl...)
Affinity DataKi:  16nMAssay Description:Inhibition of MMP2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50354624(CHEMBL1834422 | US10357546, ND-322 | US9951035, ND...)
Affinity DataKi:  24nMAssay Description:Inhibition of MMP2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))TBA
LigandPNGBDBM408486(US10357546, ND-3640)
Affinity DataKi:  40nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))TBA
LigandPNGBDBM50433867(CHEMBL2380401)
Affinity DataKi:  62nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50354625(CHEMBL1834423)
Affinity DataKi:  78nMAssay Description:Inhibition of MMP2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM408486(US10357546, ND-3640)
Affinity DataKi:  93nMAssay Description:Inhibition of MMP9 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))TBA
LigandPNGBDBM50354624(CHEMBL1834422 | US10357546, ND-322 | US9951035, ND...)
Affinity DataKi:  100nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))TBA
LigandPNGBDBM389618(US10357546, ND-336 | US9951035, ND-336 (5))
Affinity DataKi:  120nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM389618(US10357546, ND-336 | US9951035, ND-336 (5))
Affinity DataKi:  150nMAssay Description:Inhibition of MMP9 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))TBA
LigandPNGBDBM50433867(CHEMBL2380401)
Affinity DataKi:  160nMAssay Description:Inhibition of MMP12 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50610479(CHEMBL5283337)
Affinity DataKi:  180nMAssay Description:Inhibition of MMP9 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))TBA
LigandPNGBDBM50354625(CHEMBL1834423)
Affinity DataKi:  260nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50354625(CHEMBL1834423)
Affinity DataKi:  490nMAssay Description:Inhibition of MMP9 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeutrophil collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50405531(CHEMBL5270713)
Affinity DataKi:  692nMAssay Description:Inhibition of MMP8 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeutrophil collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM408486(US10357546, ND-3640)
Affinity DataKi:  730nMAssay Description:Inhibition of MMP8 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50354624(CHEMBL1834422 | US10357546, ND-322 | US9951035, ND...)
Affinity DataKi:  870nMAssay Description:Inhibition of MMP9 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrilysin(Homo sapiens (Human))TBA
LigandPNGBDBM50433864(CHEMBL2380403)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeutrophil collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM389618(US10357546, ND-336 | US9951035, ND-336 (5))
Affinity DataKi:  7.70E+3nMAssay Description:Inhibition of MMP8 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))TBA
LigandPNGBDBM50610473(CHEMBL5286645)
Affinity DataKi:  9.40E+3nMAssay Description:Inhibition of MMP14 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrilysin(Homo sapiens (Human))TBA
LigandPNGBDBM50433867(CHEMBL2380401)
Affinity DataKi: >2.50E+4nMAssay Description:Inhibition of MMP7 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50610473(CHEMBL5286645)
Affinity DataKi:  3.40E+4nMAssay Description:Inhibition of MMP9 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrilysin(Homo sapiens (Human))TBA
LigandPNGBDBM50608587(CHEMBL5274327)
Affinity DataKi:  1.16E+5nMAssay Description:Inhibition of MMP7 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50610465(CHEMBL5288452)
Affinity DataIC50:  0.0449nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50610466(CHEMBL5280430)
Affinity DataIC50:  0.0650nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50608587(CHEMBL5274327)
Affinity DataIC50:  0.220nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50610470(CHEMBL5271422)
Affinity DataIC50:  0.230nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50610466(CHEMBL5280430)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of MMP9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50610465(CHEMBL5288452)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of MMP9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))TBA
LigandPNGBDBM50610465(CHEMBL5288452)
Affinity DataIC50:  0.368nMAssay Description:Inhibition of MMP12 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))TBA
LigandPNGBDBM50610466(CHEMBL5280430)
Affinity DataIC50:  0.566nMAssay Description:Inhibition of MMP12 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNeutrophil collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50610465(CHEMBL5288452)
Affinity DataIC50:  0.567nMAssay Description:Inhibition of MMP8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM413584((2S,4R)—N-[(1S)-1-[[(1S)-3-benzamido-1-(hydro...)
Affinity DataIC50: <1nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50608587(CHEMBL5274327)
Affinity DataIC50:  1nMAssay Description:Inhibition of MMP9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50433867(CHEMBL2380401)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of MMP9 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50433864(CHEMBL2380403)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of MMP2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50433867(CHEMBL2380401)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of MMP2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50433864(CHEMBL2380403)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of MMP9 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM413584((2S,4R)—N-[(1S)-1-[[(1S)-3-benzamido-1-(hydro...)
Affinity DataIC50:  10nMAssay Description:Inhibition of MMP9 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM413580((2 S)-1-[(2S)-2-[acetyl(methyl)amino]propanoyl]-N-...)
Affinity DataIC50:  21nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand Info
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM408486(US10357546, ND-3640)
Affinity DataIC50:  21nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50610471(CHEMBL5280125)
Affinity DataIC50:  27nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50610467(CHEMBL5283653)
Affinity DataIC50:  41nMAssay Description:Inhibition of MMP9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50610467(CHEMBL5283653)
Affinity DataIC50:  50nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))TBA
LigandPNGBDBM50610467(CHEMBL5283653)
Affinity DataIC50:  50nMAssay Description:Inhibition of MMP12 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50610468(CHEMBL5281175)
Affinity DataIC50:  53nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM50610469(CHEMBL5284973)
Affinity DataIC50:  55nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))TBA
LigandPNGBDBM50264810(CHEMBL445971 | N-(4-(4-(thiiran-2-ylmethylsulfonyl...)
Affinity DataIC50:  80nMAssay Description:Inhibition of MMP9 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))TBA
LigandPNGBDBM389618(US10357546, ND-336 | US9951035, ND-336 (5))
Affinity DataIC50:  85nMAssay Description:Inhibition of MMP2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
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