Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 50033357
Affinity DataKi: 0.700nMAssay Description:Displacement of [125I]iodoproxyfan from human full-length histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]histamine from human full-length histamine H4 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [125I]iodoproxyfan from human full-length histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]histamine from human full-length histamine H4 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H]histamine from human full-length histamine H4 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [125I]iodoproxyfan from human full-length histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [125I]iodoproxyfan from human full-length histamine H3 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 154nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2 subunit after 60 mins b...More data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2 subunit after 60 mins b...More data for this Ligand-Target Pair
Affinity DataKi: 194nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 378nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2 subunit after 60 mins b...More data for this Ligand-Target Pair
Affinity DataKi: 421nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2 subunit after 60 mins b...More data for this Ligand-Target Pair
Affinity DataKi: 447nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2 subunit after 60 mins b...More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2 subunit after 60 mins b...More data for this Ligand-Target Pair
Affinity DataKi: 612nMAssay Description:Displacement of [3H]histamine from human full-length histamine H4 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
Affinity DataKi: 703nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2 subunit after 60 mins b...More data for this Ligand-Target Pair
Affinity DataKi: 1.05E+3nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2 subunit after 60 mins b...More data for this Ligand-Target Pair
Affinity DataKi: 1.33E+3nMAssay Description:Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2 subunit after 60 mins b...More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Antagonist activity against histamine H3 receptor in guinea pig ileum assessed as inhibition of electrically-evoked twitches after 30 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity against histamine H3 receptor in guinea pig ileum assessed as inhibition of electrically-evoked twitches after 30 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Antagonist activity against histamine H3 receptor in guinea pig ileum assessed as inhibition of electrically-evoked twitches after 30 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 43nMAssay Description:Antagonist activity against histamine H3 receptor in guinea pig ileum assessed as inhibition of electrically-evoked twitches after 30 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Antagonist activity against histamine H3 receptor in guinea pig ileum assessed as inhibition of electrically-evoked twitches after 30 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Antagonist activity against histamine H3 receptor in guinea pig ileum assessed as inhibition of electrically-evoked twitches after 30 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:Antagonist activity against histamine H3 receptor in guinea pig ileum assessed as inhibition of electrically-evoked twitches after 30 mins in presenc...More data for this Ligand-Target Pair
Affinity DataIC50: 128nMAssay Description:Antagonist activity against histamine H3 receptor in guinea pig ileum assessed as inhibition of electrically-evoked twitches after 30 mins in presenc...More data for this Ligand-Target Pair
Affinity DataKd: >3.02E+3nMAssay Description:Antagonist activity at histamine H1 receptor in guinea-pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+5nMAssay Description:Antagonist activity at histamine H1 receptor in guinea-pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 1.07E+4nMAssay Description:Antagonist activity at histamine H1 receptor in guinea-pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 6.92E+4nMAssay Description:Antagonist activity at histamine H1 receptor in guinea-pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 7.94E+4nMAssay Description:Antagonist activity at histamine H1 receptor in guinea-pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 4.68E+4nMAssay Description:Antagonist activity at histamine H1 receptor in guinea-pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 1.10E+5nMAssay Description:Antagonist activity at histamine H1 receptor in guinea-pig ileumMore data for this Ligand-Target Pair