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Found 2 Enz. Inhib. hit(s) with Target = '11-beta-hydroxysteroid dehydrogenase 1' and Ligand = 'BDBM50207795'
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
University Of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207795(CHEMBL246952 | adamantan-1-yl-(3,4-dihydro-2H-quin...)
Affinity DataIC50:  481nMAssay Description:Inhibition of mouse 11beta-HSD1 expressed in CHO cells after 4 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
University Of Edinburgh

Curated by ChEMBL
LigandPNGBDBM50207795(CHEMBL246952 | adamantan-1-yl-(3,4-dihydro-2H-quin...)
Affinity DataIC50:  1.86E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK293 cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed