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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50097673'
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50097673(CHEMBL3589578)
Affinity DataKi:  0.603nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A receptor by PDSP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50097673(CHEMBL3589578)
Affinity DataEC50:  10nMAssay Description:Partial agonist activity at human 5-HT2A receptor expressed in human tsA201 cells after 30 mins by inositol phosphate turnover assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed