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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50422942'
TargetAdenosine receptor A1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50422942(CHEMBL414055)
Affinity DataKd:  158nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50422942(CHEMBL414055)
Affinity DataKd:  891nMAssay Description:Binding affinity to N-terminal NLuc tagged rat A1 adenosine receptor expressed in Flp-In-CHO cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50422942(CHEMBL414055)
Affinity DataKd:  1.02E+3nMAssay Description:Binding affinity to N-terminal NLuc tagged human A1 adenosine receptor expressed in Flp-In-CHO cells by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed