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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM85776'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85776(CAS_393594 | CHEMBL89852 | MRS1191 | NSC_393594)
Affinity DataKi:  40.1nMAssay Description:Binding affinity was determined in radioligand binding assay at rat brain adenosine A1 receptor vs [3H]-R-PIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85776(CAS_393594 | CHEMBL89852 | MRS1191 | NSC_393594)
Affinity DataKi:  4.01E+4nMAssay Description:Binding affinity against adenosine A1 receptor in rat cerebral cortex membrane by radioligand binding assay using [3H](R)-PIA.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85776(CAS_393594 | CHEMBL89852 | MRS1191 | NSC_393594)
Affinity DataKi:  4.01E+4nMAssay Description:Displacement of [3H]-R-PIA from adenosine A1 receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM85776(CAS_393594 | CHEMBL89852 | MRS1191 | NSC_393594)
Affinity DataKi:  4.01E+4nMAssay Description:Displacement of specific [3H]-(R)-PIA binding at adenosine A1 receptor from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed