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Report error Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2b' and Ligand = 'BDBM50233082'
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50233082(8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50233082(8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]ZM-241385 from human recombinant adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Human)
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50233082(8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-ZM241385 from human A2B receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed