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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50078421'
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50078421(CHEMBL3414948)
Affinity DataKi:  0.588nMAssay Description:Displacement of [3H]-HEMADO from human recombinant adenosine A3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50078421(CHEMBL3414948)
Affinity DataEC50:  13nMAssay Description:Antagonist activity at human recombinant adenosine A3 receptor transfected in CHO cells assessed as reversal of NECA-induced inhibition of forskolin-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed