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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50145226'
TargetAdenosine receptor A3(Homo sapiens (Human))
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50145226(5-Butyl-2-phenyl-[1,2,4]triazolo[1,5-c]quinazoline...)
Affinity DataIC50:  260nMAssay Description:Binding affinity for human adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50145226(5-Butyl-2-phenyl-[1,2,4]triazolo[1,5-c]quinazoline...)
Affinity DataIC50:  260nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed